日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Substrate-Guided Development of HDAC11-Selective Inhibitors Featuring α‑Amino Amide Zinc-Binding Groups

基于底物导向的HDAC11选择性抑制剂的开发,该抑制剂具有α-氨基酰胺锌结合基团

Hilscher, Sebastian; Meleshin, Marat; Baselious, Fady; Barinka, Cyril; Sippl, Wolfgang; Schutkowski, Mike; Schiene-Fischer, Cordelia

Identification of Rapaglutin E as an Isoform-Specific Inhibitor of Glucose Transporter 1

雷帕格鲁汀E被鉴定为葡萄糖转运蛋白1的同工型特异性抑制剂

Kotlyar, Marnie; Guo, Zufeng; Rao, A V Subba; Peng, Hanjing; Wang, Jingxin; Ma, Zhongnan; Schiene-Fischer, Cordelia; Fischer, Gunter; Liu, Jun O

Continuous Fluorescent Sirtuin Activity Assay Based on Fatty Acylated Lysines

基于脂肪酰化赖氨酸的连续荧光 Sirtuin 活性测定

Matthes Zessin, Marat Meleshin, Sebastian Hilscher, Cordelia Schiene-Fischer, Cyril Barinka, Manfred Jung, Mike Schutkowski

Non-Immunosuppressive Cyclophilin Inhibitors

非免疫抑制性亲环蛋白抑制剂

Schiene-Fischer, Cordelia; Fischer, Gunter; Braun, Manfred

Rapamycin-inspired macrocycles with new target specificity

雷帕霉素启发的具有新型靶向特异性的大环化合物

Guo, Zufeng; Hong, Sam Y; Wang, Jingxin; Rehan, Shahid; Liu, Wukun; Peng, Hanjing; Das, Manisha; Li, Wei; Bhat, Shridhar; Peiffer, Brandon; Ullman, Brett R; Tse, Chung-Ming; Tarmakova, Zlatina; Schiene-Fischer, Cordelia; Fischer, Gunter; Coe, Imogen; Paavilainen, Ville O; Sun, Zhaoli; Liu, Jun O

Discovery of a Potent GLUT Inhibitor from a Library of Rapafucins by Using 3D Microarrays

利用三维微阵列技术从雷帕霉素库中发现强效GLUT抑制剂

Guo, Zufeng; Cheng, Zhiqiang; Wang, Jingxin; Liu, Wukun; Peng, Hanjing; Wang, Yuefan; Rao, A V Subba; Li, Ruo-Jing; Ying, Xue; Korangath, Preethi; Liberti, Maria V; Li, Yingjun; Xie, Yongmei; Hong, Sam Y; Schiene-Fischer, Cordelia; Fischer, Gunter; Locasale, Jason W; Sukumar, Saraswati; Zhu, Heng; Liu, Jun O

PrsA2 (CD630_35000) of Clostridioides difficile Is an Active Parvulin-Type PPIase and a Virulence Modulator

艰难梭菌的 PrsA2 (CD630_35000) 是一种活性 Parvulin 型 PPIase 和毒力调节因子

Ünal, Can Murat; Berges, Mareike; Smit, Nathiana; Schiene-Fischer, Cordelia; Priebe, Christina; Strowig, Till; Jahn, Dieter; Steinert, Michael

Pharmacological Cyclophilin Inhibitors Prevent Intoxication of Mammalian Cells with Bordetella pertussis Toxin

药理学环丝氨酸蛋白酶抑制剂可防止哺乳动物细胞被百日咳毒素中毒

Katharina Ernst, Nina Eberhardt, Ann-Katrin Mittler, Michael Sonnabend, Anna Anastasia, Simon Freisinger, Cordelia Schiene-Fischer, Miroslav Malešević, Holger Barth

The Hsp90 machinery facilitates the transport of diphtheria toxin into human cells

Hsp90 机制促进白喉毒素进入人体细胞。

Schuster, Manuel; Schnell, Leonie; Feigl, Peter; Birkhofer, Carina; Mohr, Katharina; Roeder, Maurice; Carle, Stefan; Langer, Simon; Tippel, Franziska; Buchner, Johannes; Fischer, Gunter; Hausch, Felix; Frick, Manfred; Schwan, Carsten; Aktories, Klaus; Schiene-Fischer, Cordelia; Barth, Holger

Hsp70 facilitates trans-membrane transport of bacterial ADP-ribosylating toxins into the cytosol of mammalian cells

Hsp70 促进细菌 ADP 核糖基化毒素跨膜运输到哺乳动物细胞的胞质溶胶

Katharina Ernst, Johannes Schmid, Matthias Beck, Marlen Hägele, Meike Hohwieler, Patricia Hauff, Anna Katharina Ückert, Anna Anastasia, Michael Fauler, Thomas Jank, Klaus Aktories, Michel R Popoff, Cordelia Schiene-Fischer, Alexander Kleger, Martin Müller, Manfred Frick, Holger Barth