日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

STING Agonist VB-85247 Induces Durable Antitumor Immune Responses by Intravesical Administration in a Non-Muscle-Invasive Bladder Cancer

STING激动剂VB-85247通过膀胱内给药,在非肌层浸润性膀胱癌中诱导持久的抗肿瘤免疫反应

Miglena G Prabagar ,Michael McQueney ,Venu Bommireddy ,Rachael Siegel ,Gary L Schieven ,Ku Lu ,Ruziboy Husanov ,Reema Deepak ,David Diller ,Chia-Yu Huang ,Eli Mordechai ,Rukiye-Nazan Eraslan

Discovery of Novel TLR7 Agonists as Systemic Agent for Combination With aPD1 for Use in Immuno-oncology

发现新型TLR7激动剂作为全身性药物与抗PD-1抗体联合用于免疫肿瘤学

Poudel, Yam B; He, Liqi; Cox, Matthew; Zhang, Qian; Johnson, Walter L; Cong, Qiang; Cheng, Heng; Chowdari, Naidu S; Tarby, Christine; Donnell, Andrew F; Broekema, Matthais; O'Malley, Daniel P; Zhang, Yong; A M Subbaiah, Murugaiah; Kumar, Boda Vijay; Subramani, Lakshumanan; Wang, Bei; Li, Yi-Xin; Sivaprakasam, Prasanna; Critton, David; Mulligan, Dawn; Sandhu, Bhupindar; Xie, Chunshan; Ramakrishnan, Radha; Nagar, Jignesh; Dudhgaonkar, Shailesh; Oderinde, Martins S; Murtaza, Anwar; Schieven, Gary L; Mathur, Arvind; Gavai, Ashvinikumar V; Vite, Gregory; Gangwar, Sanjeev

Identification and Optimization of Small Molecule Pyrazolopyrimidine TLR7 Agonists for Applications in Immuno-oncology

鉴定和优化小分子吡唑并嘧啶类TLR7激动剂在免疫肿瘤学中的应用

He, Liqi; Zhang, Meng Yao; Cox, Matthew; Zhang, Qian; Donnell, Andrew F; Zhang, Yong; Tarby, Christine; Gill, Patrice; Subbaiah, Murugaiah A M; Ramar, Thangeswaran; Reddy, Maheswara; Puttapaka, Vijaya; Li, Yi-Xin; Sivaprakasam, Prasanna; Critton, David; Mulligan, Dawn; Xie, Chunshan; Ramakrishnan, Radha; Nagar, Jignesh; Dudhgaonkar, Shailesh; Murtaza, Anwar; Oderinde, Martins S; Schieven, Gary L; Mathur, Arvind; Gavai, Ashvinikumar V; Vite, Gregory; Gangwar, Sanjeev; Poudel, Yam B

An adverse tumor-protective effect of IDO1 inhibition

IDO1抑制的不良肿瘤保护作用

Juliana C N Kenski,Xinyao Huang,David W Vredevoogd,Beaunelle de Bruijn,Joleen J H Traets,Sofía Ibáñez-Molero,Sebastiaan M Schieven,Alex van Vliet,Oscar Krijgsman,Thomas Kuilman,Joanna Pozniak,Fabricio Loayza-Puch,Alexandra M Terry,Judith Müller,Meike E W Logtenberg,Marjolein de Bruijn,Pierre Levy,Pierre-René Körner,Colin R Goding,Ton N Schumacher,Jean-Christophe Marine,Reuven Agami,Daniel S Peeper

The Elongin BC Complex Negatively Regulates AXL and Marks a Differentiated Phenotype in Melanoma

Elongin BC 复合物负向调控 AXL 并标记黑色素瘤的分化表型

Sebastiaan M Schieven, Joleen J H Traets, Alex V Vliet, Martijn V Baalen, Ji-Ying Song, Marcos Da Silva Guimaraes, Thomas Kuilman, Daniel S Peeper

1049. Outcome and Impact of Empirical Antimicrobial Treatment in Bacteraemia With Bacteroides Species; A Retrospective Cohort Study in a Region of Southern Sweden

1049. 瑞典南部地区一项回顾性队列研究:拟杆菌属菌血症经验性抗菌治疗的疗效和影响

Stoakes, L; Kelly, T; Manarin, K; Schieven, B; Lannigan, R; Groves, D; Hussain, Z; Tham, Johan; Kalin, Karolina; Resman, Fredrik; Holm, Karin

Novel lung imaging biomarkers and skin gene expression subsetting in dasatinib treatment of systemic sclerosis-associated interstitial lung disease

达沙替尼治疗系统性硬化症相关间质性肺疾病中的新型肺部影像生物标志物和皮肤基因表达亚组分析

Martyanov, Viktor; Kim, Grace-Hyun J; Hayes, Wendy; Du, Shuyan; Ganguly, Bishu J; Sy, Oumar; Lee, Sun Ku; Bogatkevich, Galina S; Schieven, Gary L; Schiopu, Elena; Marangoni, Roberta Gonçalves; Goldin, Jonathan; Whitfield, Michael L; Varga, John

Homer1/mGluR5 activity moderates vulnerability to chronic social stress

Homer1/mGluR5 活性可减轻慢性社会压力的脆弱性

Klaus V Wagner, Jakob Hartmann, Christiana Labermaier, Alexander S Häusl, Gengjing Zhao, Daniela Harbich, Bianca Schmid, Xiao-Dong Wang, Sara Santarelli, Christine Kohl, Nils C Gassen, Natalie Matosin, Marcel Schieven, Christian Webhofer, Christoph W Turck, Lothar Lindemann, Georg Jaschke, Joseph G

Assessing behavioural effects of chronic HPA axis activation using conditional CRH-overexpressing mice

利用条件性CRH过表达小鼠评估慢性HPA轴激活的行为效应

Dedic, Nina; Touma, Chadi; Romanowski, Cristoph P; Schieven, Marcel; Kühne, Claudia; Ableitner, Martin; Lu, Ailing; Holsboer, Florian; Wurst, Wolfgang; Kimura, Mayumi; Deussing, Jan M

Dasatinib, a small-molecule protein tyrosine kinase inhibitor, inhibits T-cell activation and proliferation

达沙替尼是一种小分子蛋白酪氨酸激酶抑制剂,可抑制 T 细胞活化和增殖

Andrew E Schade, Gary L Schieven, Robert Townsend, Anna M Jankowska, Vojkan Susulic, Rosemary Zhang, Hadrian Szpurka, Jaroslaw P Maciejewski