日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Controlled human infection with Mycobacterium tuberculosis: practical considerations for clinical trials

控制性人体结核分枝杆菌感染:临床试验的实用性考量

Seshadri, Chetan; Flynn, JoAnne L; Maiello, Pauline; Schnappinger, Dirk; Wilkinson, Robert J; Gordon, Stephen B; Mwandumba, Henry C; Jambo, Kondwani C; Hoft, Daniel F; Rubin, Eric J; Jamrozik, Euzebiusz; Fortune, Sarah M; Kublin, James G

Activation of L-histidine biosynthesis as a new antibiotic strategy against Mycobacterium tuberculosis

激活L-组氨酸生物合成作为对抗结核分枝杆菌的新型抗生素策略

Hunt, Debbie M; Pisco, João Pedro; Rodgers, Angela; de Chiara, Cesira; Zaveri, Anisha; Pacholarz, Kamila L; Evangelopoulos, Dimitrios; Garza-Garcia, Acely; Ehrt, Sabine; Schnappinger, Dirk; Barran, Perdita E; Gutierrez, Maximiliano G; de Carvalho, Luiz Pedro S

A periplasmic protein complex mediates arabinofuranosyltransferase activity and intrinsic drug resistance in Mycobacterium tuberculosis

周质蛋白复合物介导结核分枝杆菌的阿拉伯呋喃糖基转移酶活性和内在耐药性

Klevorn, Thaís; Brown, Christopher; Hardy, Christine D; Cuthbert, Bonnie J; Spencer, Amanda; Jinich, Adrián; Chan, Luming; Angala, Shiva K; Manzer, Jordan; Mendoza, Jessica; de Miranda, Rodger; Kim, Heather; Schnappinger, Dirk; Jackson, Mary; Rhee, Kyu; Goulding, Celia W; Ehrt, Sabine

Identification and Evaluation of dibasic piperidines as novel cell wall inhibitors against Mycobacterium tuberculosis

鉴定和评价二元哌啶类化合物作为新型抗结核分枝杆菌细胞壁抑制剂

Naylor, Claire; Prosser, Gareth A; Bayliss, Tracy; Berle, Lila; Wallach, Joshua B; Kim, Heather; Olvera, Rodrigo Aguilera; Thompson, Stephen; Ioerger, Thomas R; Simpson, Laura; Casanueva, Ruth; Guijarro-Lopez, Laura; Read, Kevin D; Wyatt, Paul G; Schnappinger, Dirk; Barry, Clifton E; Green, Simon R; Boshoff, Helena I; Cleghorn, Laura A T

SuFEx-based antitubercular compound irreversibly inhibits Pks13

基于 SuFEx 的抗结核化合物不可逆地抑制 Pks13

Krieger, Inna V; Sukheja, Paridhi; Yang, Baiyuan; Tang, Su; Selle, Daniel; Woods, Ashley; Engelhart, Curtis; Kumar, Pradeep; Harbut, Michael B; Liu, Dongdong; Tsuda, Brendan; Qin, Bo; Bare, Grant A L; Li, Gencheng; Chi, Victor; Gambacurta, Julian; Hvizdos, Janine; Reagan, Matthew; Jones, Isabelle L; Massoudi, Lisa M; Woolhiser, Lisa K; Cascioferro, Alessandro; Kundrick, Erica; Singh, Parul; Reiley, William; Ioerger, Thomas R; Kandula, Dilipkumar Reddy; McCabe, Jacob W; Guo, Taijie; Alland, David; Boshoff, Helena I; Schnappinger, Dirk; Robertson, Gregory T; Mdluli, Khisi; Lee, Kyoung-Jin; Dong, Jiajia; Li, Shuangwei; Schultz, Peter G; Joseph, Sean B; Love, Melissa S; Sharpless, K Barry; Petrassi, H Michael; Chatterjee, Arnab K; Sacchettini, James C; McNamara, Case W

A BCG kill switch strain protects against Mycobacterium tuberculosis in mice and non-human primates with improved safety and immunogenicity.

卡介苗杀灭开关菌株能够提高小鼠和非人灵长类动物对结核分枝杆菌的安全性和免疫原性。

Smith Alexander A, Su Hongwei, Wallach Joshua, Liu Yao, Maiello Pauline, Borish H Jacob, Winchell Caylin, Simonson Andrew W, Lin Philana Ling, Rodgers Mark, Fillmore Daniel, Sakal Jennifer, Lin Kan, Vinette Valerie, Schnappinger Dirk, Ehrt Sabine, Flynn JoAnne L

Reference-based chemical-genetic interaction profiling to elucidate small molecule mechanism of action in Mycobacterium tuberculosis

基于参考序列的化学-遗传相互作用分析阐明结核分枝杆菌中小分子的作用机制

Bond, Austin N; Orzechowski, Marek; Zhang, Shuting; Ben-Zion, Ishay; Lemmer, Allison; Garry, Nathaniel; Lee, Katie; Chen, Michael; Delano, Kayla; Gath, Emily; Golas, A Lorelei; Nietupski, Raymond; Fitzgerald, Michael; Ehrt, Sabine; Rubin, Eric J; Sassetti, Christopher M; Schnappinger, Dirk; Shoresh, Noam; Hunt, Diana K; Gomez, James E; Hung, Deborah T

Tailored phenyl ureas eradicate drug-resistant Mycobacterium tuberculosis by targeting mycolic acid cell wall assembly

定制的苯脲类化合物通过靶向分枝菌酸细胞壁组装来根除耐药结核分枝杆菌。

Mostert, Dietrich; Braun, Josef; Zimmerman, Matthew D; Engelhart, Curtis A; Berndl, Sara; Quoika, Patrick K; Kany, Andreas M; Proietto, Julianna; Penalva-Lopez, Suyapa; Wallach, Joshua B; Hirsch, Anna K H; Zacharias, Martin; Schnappinger, Dirk; Dartois, Véronique; Sieber, Stephan A

Design and Development of Lysyl tRNA Synthetase Inhibitors, for the Treatment of Tuberculosis

赖氨酰tRNA合成酶抑制剂的设计与开发,用于治疗结核病

Davis, Susan H; Mathieson, Michael; Buchanan, Kirsteen I; Dawson, Alice; Smith, Alasdair; Cocco, Mattia; Tamaki, Fabio K; Post, John M; Baragaña, Beatriz; Jansen, Chimed; Kiczun, Michael; Zuccotto, Fabio; Wood, Gavin; Scullion, Paul; Ray, Peter C; Epemolu, Ola; Lopez-Román, Eva Maria; López, Laura Guijarro; Engelhart, Curtis A; Kim, Jia; Pino, Paula A; Schnappinger, Dirk; Read, Kevin D; Encinas, Lourdes; Bates, Robert H; Wyatt, Paul G; Green, Simon R; Cleghorn, Laura A T

Design, Synthesis, and Biological Evaluation of Mono- and Diamino-Substituted Squaramide Derivatives as Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthase

单氨基和二氨基取代的方酰胺衍生物作为结核分枝杆菌腺苷三磷酸(ATP)合成酶的强效抑制剂的设计、合成和生物学评价

Palme, Paul R; Grover, Shipra; Abdelaziz, Rana; Mann, Lea; Kany, Andreas M; Ouologuem, Lina; Bartel, Karin; Sonnenkalb, Lindsay; Reiling, Norbert; Hirsch, Anna K H; Schnappinger, Dirk; Rubinstein, John L; Imming, Peter; Richter, Adrian