日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

New N-Heterocyclic Carbene Gold and Platinum Complexes with 1,3-Dialkyl-4-anisyl-5-(4-chlorophenyl)imidazol-2-ylidene Ligands for the Treatment of Esophageal Adenocarcinoma.

新型 N-杂环卡宾金铂配合物与 1,3-二烷基-4-茴香基-5-(4-氯苯基)咪唑-2-亚基配体用于治疗食管腺癌。

Ghosh Hindole, Rehm Tobias, Bhattacharyya Sangita, Lee Miru, Veeragoni Dileepkumar, Schobert Rainer, Biersack Bernhard, Dandawate Prasad

Antiparasitic and Antifungal Activities of Cetyl-Maritima, a New N-Cetyl-Modified Maritima Derivative

鲸蜡基-海藻素(一种新型N-鲸蜡基修饰的海藻素衍生物)的抗寄生虫和抗真菌活性

Al Nasr, Ibrahim S; Ma, Jingyi; Khan, Tariq A; Koko, Waleed S; Ben Abdelmalek, Imen; Schobert, Rainer; van de Sande, Wendy; Biersack, Bernhard

Antiparasitic Activities of Acyl Hydrazones from Cinnamaldehydes and Structurally Related Fragrances

肉桂醛及其结构相关香料的酰腙的抗寄生虫活性

Al Nasr, Ibrahim S; Koko, Waleed S; Khan, Tariq A; Schobert, Rainer; Biersack, Bernhard

Formal synthesis of kibdelomycin and derivatisation of amycolose glycosides

kibdelomycin 的形式合成及阿米可洛糖苷的衍生化

Schriefer, Manuel G; Treiber, Laura; Schobert, Rainer

Multimodal 4-arylchromene derivatives with microtubule-destabilizing, anti-angiogenic, and MYB-inhibitory activities

具有微管解聚、抗血管生成和MYB抑制活性的多模式4-芳基色烯衍生物

Köhler, Leonhard H F; Reich, Sebastian; Yusenko, Maria; Klempnauer, Karl-Heinz; Begemann, Gerrit; Schobert, Rainer; Biersack, Bernhard

Antiparasitic Activity of Fluorophenyl-Substituted Pyrimido[1,2-a]benzimidazoles

氟苯基取代的嘧啶并[1,2-a]苯并咪唑的抗寄生虫活性

Nasr, Ibrahim S Al; Koko, Waleed S; Khan, Tariq A; Schobert, Rainer; Biersack, Bernhard

2-Amino-4-aryl-5-oxo-4,5-dihydropyrano[3,2-c]chromene-3-carbonitriles with Microtubule-Disruptive, Centrosome-Declustering, and Antiangiogenic Effects in vitro and in vivo

2-氨基-4-芳基-5-氧代-4,5-二氢吡喃并[3,2-c]色烯-3-腈类化合物在体外和体内均表现出微管破坏、中心体解聚和抗血管生成作用

Köhler, Leonhard H F; Reich, Sebastian; Begemann, Gerrit; Schobert, Rainer; Biersack, Bernhard

3D cell cultures, as a surrogate for animal models, enhance the diagnostic value of preclinical in vitro investigations by adding information on the tumour microenvironment: a comparative study of new dual-mode HDAC inhibitors

3D细胞培养作为动物模型的替代方法,通过提供肿瘤微环境信息,增强了临床前体外研究的诊断价值:新型双模式HDAC抑制剂的比较研究

Bär, Sofia I; Biersack, Bernhard; Schobert, Rainer

Imidazole Analogs of Vascular-Disrupting Combretastatin A-4 with Pleiotropic Efficacy against Resistant Colorectal Cancer Models

具有多效性疗效的血管破坏性康布瑞他汀A-4咪唑类似物对抗耐药性结直肠癌模型

Reipsch, Franziska; Biersack, Bernhard; Lucas, Henrike; Schobert, Rainer; Mueller, Thomas

A New Pentafluorothio-Substituted Curcuminoid with Superior Antitumor Activity

一种新型五氟硫代取代的姜黄素类化合物具有优异的抗肿瘤活性

Linder, Benedikt; Köhler, Leonhard H F; Reisbeck, Lisa; Menger, Dominic; Subramaniam, Dharmalingam; Herold-Mende, Christel; Anant, Shrikant; Schobert, Rainer; Biersack, Bernhard; Kögel, Donat