1- O-Octadecyl-2- O-benzyl- sn-glyceryl-3- phospho-GS-441524 (V2043). Evaluation of Oral V2043 in a Mouse Model of SARS-CoV-2 Infection and Synthesis and Antiviral Evaluation of Additional Phospholipid Esters with Enhanced Anti-SARS-CoV-2 Activity
1- O-十八烷基-2- O-苄基-sn-甘油基-3-磷酸-GS-441524 (V2043)。在 SARS-CoV-2 感染的小鼠模型中口服 V2043 的评估以及具有增强的抗 SARS-CoV-2 活性的其他磷脂酯的合成和抗病毒评估
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.3c00046
Aaron F Carlin, James R Beadle, Alex E Clark, Kendra L Gully, Fernando R Moreira, Ralph S Baric, Rachel L Graham, Nadejda Valiaeva, Sandra L Leibel, William Bray, Rachel E McMillan, Jonathan E Freshman, Aaron F Garretson, Rachael N McVicar, Tariq Rana, Xing-Quan Zhang, Joyce A Murphy, Robert T Schoo