日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Subtype-selective positron emission tomography imaging of poly ADP-ribose polymerase-1 binding in non-human primates, healthy volunteers, and patients with glioblastoma using [11C]AZ14193391

利用[11C]AZ14193391对非人灵长类动物、健康志愿者和胶质母细胞瘤患者进行亚型选择性正电子发射断层扫描成像,以检测聚ADP核糖聚合酶-1的结合情况。

Cselényi, Zsolt; Jucaite, Aurelija; Stragliotto, Giuseppe; Bartek, Jiri; Johnström, Peter; Pike, Andy; Cortés González, Miguel A; Högnäsbacka, Antonia; Dahl, Kenneth; Ghosh, Avipsa; Johannes, Jeffrey W; Staniszewska, Anna D; Leo, Elisabetta; Hamerlik, Petra; Davies, Barry; Cosulich, Sabina; Swales, John; Lawrence, Rachel; Squatrito, Massimo; Mueller, Nancy Kathryn; Khani, Yasir; Sousa, Vasco C; Stenkrona, Per; Halldin, Christer; Farde, Lars; Schou, Magnus

AZ14289671 is a highly selective and blood-brain barrier penetrant irreversible TKI that targets EGFRExon20 insertions.

AZ14289671 是一种高选择性且能穿透血脑屏障的不可逆 TKI,靶向 EGFRExon20 插入

Swaih Aisha M, Talbot Sara, Savoca Adriana, Thorpe Hannah, Flemington Vikki, Phillips Benjamin, Colclough Nicola, McCoull William, Radeva Veronika, Hargreaves David, Packer Martin J, Felisberto-Rodrigues Catarina, Thomson Clare, Orme Jonathan P, Deane Carly, Smith Aaron, Johnström Peter, Schou Magnus, McWilliams Lisa, Davey Paul, Enget Marianne, O'Neill Daniel, Cosulich Sabina, Floc'h Nicolas

Radiolabeling and Preliminary In Vivo Evaluation of the Candidate CCR2 Targeting PET Radioligand [(11)C]AZD2423

候选 CCR2 靶向 PET 放射性配体 [(11)C]AZD2423 的放射性标记和初步体内评价

Dahl, Kenneth; Johnström, Peter; Tóth, Miklós; Bolin, Martin; Varnäs, Katarina; Nakao, Ryuji; Takano, Akihiro; Khani Meynaq, Yasir; Bayrakdarian, Malken; Cselényi, Zsolt; Halldin, Christer; Farde, Lars; Schou, Magnus

Brain exposure of the mesenchymal-epithelial transition inhibitor savolitinib in nonhuman primates: A positron emission tomography study

非人灵长类动物脑部暴露于间质-上皮转化抑制剂萨沃替尼的情况:一项正电子发射断层扫描研究

Johnström, Peter; Cselényi, Zsolt; Miah, Kowser; Jucaite, Aurelija; Scarfe, Graeme; Cortés González, Miguel A; Farde, Lars; Halldin, Christer; Vishwanathan, Karthick; Schou, Magnus

Radiosynthesis and Evaluation of (11)C‑Labeled Imidazolyl Pyrimidine Derivatives for Positron Emission Tomography Imaging of Glycogen Synthase Kinase‑3

利用放射合成和评价(11)C标记的咪唑基嘧啶衍生物对糖原合成酶激酶-3进行正电子发射断层扫描成像

Li, Yinlong; Dahl, Kenneth; Elmore, Charles S; Sandell, Johan; Takano, Akihiro; Halldin, Christer; Farde, Lars; Ahlgren, Charlotte; Cochrane, Alison; Rong, Jian; Chen, Jiahui; Zhao, Chunyu; Zhou, Xin; Patel, Jimmy S; Song, Zhendong; Chaudhary, Ahmad; Gao, Yabiao; Sun, Zhenkun; Zhang, Zachary; Feng, Siyan; Haider, Achi; Liang, Steven H; Schou, Magnus

Re-PERFUSE: Phase 1b study of AZD3427, a novel relaxin receptor agonist, on renal perfusion in HFrEF patients

Re-PERFUSE:AZD3427(一种新型松弛素受体激动剂)对射血分数降低型心力衰竭(HFrEF)患者肾脏灌注的1b期研究

Ufnal, Marcin; Quintana-Hayashi, Macarena P; Connolly, Kathleen; Pettersen, Daniel; Cselényi, Zsolt; Jucaite, Aurelija; Schou, Magnus; Varrone, Andrea; Chan, Melanie; Lund, Lars H

PET imaging of mitochondrial complex-I in the adenine-induced tubulointerstitial nephropathy mouse model using [(18)F]BCPP-BF

利用[(18)F]BCPP-BF对腺嘌呤诱导的肾小管间质性肾病小鼠模型中的线粒体复合物I进行PET成像

Dahl, Kenneth; Johnström, Peter; Toth, Miklós; Sousa, Vasco C; Ericsson, Charlotte; Strömstedt, Maria; Inghardt, Tord; Cortés González, Miguel A; Reznichenko, Anna; Jucaite, Aurelija; Cselényi, Zsolt; Unwin, Robert; Ohba, Hiroyuki; Halldin, Christer; Challis, Benjamin; Tsukada, Hideo; Schou, Magnus

Identification and In Vitro and In Vivo Characterization of KAC-50.1 as a Potential α-Synuclein PET Radioligand

KAC-50.1作为潜在的α-突触核蛋白PET放射性配体的鉴定、体外和体内表征

Saturnino Guarino, Dinahlee; Miranda Azpiazu, Patricia; Sunnemark, Dan; Elmore, Charles S; Bergare, Jonas; Artelsmair, Markus; Nordvall, Gunnar; Forsberg Morén, Anton; Jia, Zhisheng; Cortes-Gonzalez, Miguel; Mach, Robert H; Wilcox, Kyle C; Finnema, Sjoerd; Schou, Magnus; Varrone, Andrea

Radiosynthesis and Evaluation of 11C-Labeled Isoindolone-Based Positive Allosteric Modulators for Positron Emission Tomography Imaging of Metabotropic Glutamate Receptor 2

利用 11C 标记的异吲哚酮类正变构调节剂进行放射合成和评价,用于代谢型谷氨酸受体 2 的正电子发射断层扫描成像

Li, Yinlong; Dahl, Kenneth; Johnström, Peter; Varnäs, Katarina; Farde, Lars; Halldin, Christer; Medd, Amy; Maier, Donna; Powell, Mark E; Chen, Jiahui; Van, Richard; Patel, Jimmy; Chaudhary, Ahmad; Gao, Yabiao; Song, Zhendong; Haider, Achi; Shao, Yihan; Elmore, Charles S; Liang, Steven; Schou, Magnus

Reactive Palladium-Ligand Complexes for (11)C-Carbonylation at Ambient Pressure: A Breakthrough in Carbon-11 Chemistry

常压下用于 (11)C-羰基化的活性钯-配体配合物:碳-11化学的突破

Dahl, Kenneth; Lindberg, Anton; Vasdev, Neil; Schou, Magnus