日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Advanced Molecular Tweezers Effectively Target Membranes Lacking Choline Headgroups for Broad-Spectrum Antiviral Efficacy

先进的分子镊子可有效靶向缺乏胆碱头基的细胞膜,从而实现广谱抗病毒疗效

Weil, Tatjana; Lawrenz, Jan; Taghuo Kaptouom, Estelle; Mieres-Perez, Joel; Hunszinger, Victoria; Sparrer, Konstantin M J; Almeida-Hernandez, Yasser; Schrader, Thomas; Sanchez-Garcia, Elsa; Münch, Jan

Allosteric Modulation of Pathological Ataxin-3 Aggregation: A Path to Spinocerebellar Ataxia Type-3 Therapies

病理性共济蛋白-3聚集的变构调节:脊髓小脑性共济失调3型治疗的途径

Silva, Alexandra; Duarte-Silva, Sara; Martins, Pedro M; Rodrigues, Beatriz; Serrenho, Débora; Vilasboas-Campos, Daniela; Teixeira-Castro, Andreia; Vieyto-Nuñez, Julio; Mieres-Perez, Joel; Figueiredo, Francisco; Podlasiak, Martyna; Van-der-Kellen, Tatiana; Fraga, Joana; Noble, James; Lantz, Carter; Sepanj, Niki; Monteiro-Fernandes, Daniela; Guerreiro, Sara; Neves-Carvalho, Andreia; Pereira-Sousa, Joana; Klärner, Frank-Gerrit; Schrader, Thomas; Loo, Joseph A; Pastore, Annalisa; Sanchez-Garcia, Elsa; Bitan, Gal; Carvalho, Ana Luísa; Maciel, Patrícia; Macedo-Ribeiro, Sandra

Molecular tweezer-peptide conjugates disrupt the protein-protein interaction between survivin and histone H3 essential in mitosis

分子镊子-肽缀合物破坏了存活蛋白和组蛋白H3之间在有丝分裂中至关重要的蛋白质-蛋白质相互作用

Gsell, Catherine; Rebmann, Philipp; Opara, Karina; Beuck, Christine; Bayer, Peter; Bier, David; Vetter, Ingrid R; Schrader, Thomas

Molecular Tweezers Block the Functional Pore of a Protein Machine

分子镊子阻断蛋白质机器的功能孔

Kirupakaran, Abbna; van den Boom, Johannes; Blueggel, Mike; Beuck, Christine; Niemeyer, Felix; Hayduk, Matthias; Balszuweit, Jan; Bayer, Peter; Voskuhl, Jens; Meyer, Hemmo; Schrader, Thomas

Diazepine Agonists of the 5-HT(2C) Receptor with Unprecedented Selectivity: Discovery of Bexicaserin (LP352)

具有前所未有的选择性的 5-HT(2C) 受体二氮卓类激动剂:Bexicaserin (LP352) 的发现

Ren, Albert; Zhu, Xiuwen; Lehmann, Juerg; Kasem, Michelle; Schrader, Thomas O; Dang, Huong; Le, Minh; Frazer, John; Unett, David J; Grottick, Andrew J; Whelan, Kevin T; Morgan, Michael E; Sage, Carleton R; Srinivas, Nuggehally R; McLin, Dewey; Semple, Graeme

The LPAR1 antagonist, PIPE-791 produces antifibrotic effects in models of lung fibrosis

LPAR1拮抗剂PIPE-791在肺纤维化模型中产生抗纤维化作用

Poon, Michael; Lorrain, Kym; Broadhead, Alexander; Stebbins, Karin; Bagnol, Didier; Edu, Geraldine; Joseph, Gregory; Baccei, Christopher; Roppe, Jeffrey; Schrader, Thomas; Valdez, Lino; Xiong, Yifeng; Chen, Austin; Lorrain, Daniel

Photoresponsive molecular tweezers modulate Taspase 1 activity

光响应分子镊子调节Taspase 1活性

Bietti, Antonio L Figueroa; Kauth, Alisa-Maite A; Hommel, Katrin; Blueggel, Mike; Mohr, Laurenz; Niemeyer, Felix C; Beuck, Christine; Bayer, Peter; Knauer, Shirley K; Jan Ravoo, Bart; Schrader, Thomas

Monitoring Receptor Clustering by Aggregation-Induced Emission

通过聚集诱导发射监测受体聚集

Bekus, Robert; Rudolph, Kevin; Riebe, Steffen; Voskuhl, Jens; Schrader, Thomas

Strategic implementation of HPV vaccination to eliminate cervical cancer in Georgia

在格鲁吉亚战略性地实施HPV疫苗接种,以消除宫颈癌

Khuntsaria, Irakli; Gachechiladze, Konstantine; Liparta, Elene; Kobulashvili, Tamar; Jorbenadze, Mariam; Revazishvili, Tamaz; Mamiseishvili, Ana; Kekelia, Elene; Topuridze, Marina; Sturua, Lela; Schrader, Thomas; Kldiashvili, Ekaterina

How Do Molecular Tweezers Bind to Proteins? Lessons from X-ray Crystallography

分子镊子如何与蛋白质结合?来自X射线晶体学的启示

Porfetye, Arthur T; Stege, Patricia; Rebollido-Rios, Rocio; Hoffmann, Daniel; Schrader, Thomas; Vetter, Ingrid R