日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An Ultra-High-Throughput Screen for Catalytic Inhibitors of Serine/Threonine Protein Phosphatases Types 1 and 5 (PP1C and PP5C)

丝氨酸/苏氨酸蛋白磷酸酶1型和5型(PP1C和PP5C)催化抑制剂的超高通量筛选

Swingle, Mark; Volmar, Claude-Henry; Saldanha, S Adrian; Chase, Peter; Eberhart, Christina; Salter, Edward A; D'Arcy, Brandon; Schroeder, Chad E; Golden, Jennifer E; Wierzbicki, Andrzej; Hodder, Peter; Honkanen, Richard E

Crystal structures and mutagenesis of PPP-family ser/thr protein phosphatases elucidate the selectivity of cantharidin and novel norcantharidin-based inhibitors of PP5C.

PPP家族丝氨酸/苏氨酸蛋白磷酸酶的晶体结构和诱变研究阐明了斑蝥素和新型去甲斑蝥素类PP5C抑制剂的选择性

Chattopadhyay Debasish, Swingle Mark R, Salter Edward A, Wood Eric, D'Arcy Brandon, Zivanov Catherine, Abney Kevin, Musiyenko Alla, Rusin Scott F, Kettenbach Arminja, Yet Larry, Schroeder Chad E, Golden Jennifer E, Dunham Wade H, Gingras Anne-Claude, Banerjee Surajit, Forbes David, Wierzbicki Andrzej, Honkanen Richard E

Discovery of a Broad-Spectrum Antiviral Compound That Inhibits Pyrimidine Biosynthesis and Establishes a Type 1 Interferon-Independent Antiviral State

发现一种广谱抗病毒化合物,该化合物可抑制嘧啶生物合成并建立一种不依赖于I型干扰素的抗病毒状态

Chung, Dong-Hoon; Golden, Jennifer E; Adcock, Robert S; Schroeder, Chad E; Chu, Yong-Kyu; Sotsky, Julie B; Cramer, Daniel E; Chilton, Paula M; Song, Chisu; Anantpadma, Manu; Davey, Robert A; Prodhan, Aminul I; Yin, Xinmin; Zhang, Xiang

Development of (E)-2-((1,4-dimethylpiperazin-2-ylidene)amino)-5-nitro-N-phenylbenzamide, ML336: Novel 2-amidinophenylbenzamides as potent inhibitors of venezuelan equine encephalitis virus

(E)-2-((1,4-二甲基哌嗪-2-亚基)氨基)-5-硝基-N-苯基苯甲酰胺,ML336 的开发:新型 2-脒基苯基苯甲酰胺类化合物作为委内瑞拉马脑炎病毒的强效抑制剂

Schroeder, Chad E; Yao, Tuanli; Sotsky, Julie; Smith, Robert A; Roy, Sudeshna; Chu, Yong-Kyu; Guo, Haixun; Tower, Nichole A; Noah, James W; McKellip, Sara; Sosa, Melinda; Rasmussen, Lynn; Smith, Layton H; White, E Lucile; Aubé, Jeffrey; Jonsson, Colleen B; Chung, Donghoon; Golden, Jennifer E

Optimization of potent and selective quinazolinediones: inhibitors of respiratory syncytial virus that block RNA-dependent RNA-polymerase complex activity.

优化高效选择性喹唑啉二酮类化合物:呼吸道合胞病毒抑制剂,可阻断 RNA 依赖性 RNA 聚合酶复合物的活性

Matharu Daljit S, Flaherty Daniel P, Simpson Denise S, Schroeder Chad E, Chung Donghoon, Yan Dan, Noah James W, Jonsson Colleen B, White E Lucile, Aubé Jeffrey, Plemper Richard K, Severson William E, Golden Jennifer E

Ebselen inhibits hepatitis C virus NS3 helicase binding to nucleic acid and prevents viral replication.

依布硒能抑制丙型肝炎病毒 NS3 解旋酶与核酸的结合,从而阻止病毒复制

Mukherjee Sourav, Weiner Warren S, Schroeder Chad E, Simpson Denise S, Hanson Alicia M, Sweeney Noreena L, Marvin Rachel K, Ndjomou Jean, Kolli Rajesh, Isailovic Dragan, Schoenen Frank J, Frick David N

Interrogating a hexokinase-selected small-molecule library for inhibitors of Plasmodium falciparum hexokinase

筛选己糖激酶筛选的小分子化合物库,以寻找恶性疟原虫己糖激酶抑制剂

Harris, Michael T; Walker, Dawn M; Drew, Mark E; Mitchell, William G; Dao, Kevin; Schroeder, Chad E; Flaherty, Daniel P; Weiner, Warren S; Golden, Jennifer E; Morris, James C

Tax protein-induced expression of antiapoptotic Bfl-1 protein contributes to survival of human T-cell leukemia virus type 1 (HTLV-1)-infected T-cells

Tax蛋白诱导的抗凋亡蛋白Bfl-1的表达有助于人类T细胞白血病病毒1型(HTLV-1)感染的T细胞的存活。

Zhang, Yi-Ya; Huang, Yong; He, Quan-Ze; Luo, Ji; Zhu, Li; Lu, Shan-Shan; Liu, Jin-Yan; Huang, Peng-Fei; Zeng, Xiong-Zhi; Liang, Song-Ping; Zhao, Peishen; Lieu, TinaMarie; Barlow, Nicholas; Metcalf, Matthew; Veldhuis, Nicholas; Jensen, Dane D; Kocan, Martina; Sostegni, Silvia; Haerteis, Silke; Baraznenok, Vera; Henderson, Ian; Lindström, Erik; Guerrero-Alba, Raquel; Valdez-Morales, Eduardo E; Liedtke, Wolfgang; McIntyre, Peter; Vanner, Stephen J; Korbmacher, Christoph; Bunnett, Nigel W; Pero, Raffaela; Palmieri, Dario; Angrisano, Tiziana; Valentino, Teresa; Federico, Antonella; Franco, Renato; Lembo, Francesca; Klein-Szanto, Andres J; Del Vecchio, Luigi; Montanaro, Donatella; Keller, Simona; Arra, Claudio; Papadopoulou, Vasiliki; Wagner, Simon D; Croce, Carlo M; Fusco, Alfredo; Chiariotti, Lorenzo; Fedele, Monica; Hong, Lin; Kenney, S Ray; Phillips, Genevieve K; Simpson, Denise; Schroeder, Chad E; Nöth, Julica; Romero, Elsa; Swanson, Scarlett; Waller, Anna; Strouse, J Jacob; Carter, Mark; Chigaev, Alexandre; Ursu, Oleg; Oprea, Tudor; Hjelle, Brian; Golden, Jennifer E; Aubé, Jeffrey; Hudson, Laurie G; Buranda, Tione; Sklar, Larry A; Wandinger-Ness, Angela; Yongqing, Tang; Wilmann, Pascal G; Reeve, Shane B; Coetzer, Theresa H; Smith, A Ian; Whisstock, James C; Pike, Robert N; Wijeyewickrema, Lakshmi C; Shilling, Dustin; Foskett, J Kevin; Marchant, Jan; Cowper, Ben; Liu, Yan; Lai, Livia; Pinzan, Camila; Marq, Jean Baptiste; Friedrich, Nikolas; Sawmynaden, Kovilen; Liew, Lloyd; Chai, Wengang; Childs, Robert A; Saouros, Savvas; Simpson, Peter; Roque Barreira, Maria Cristina; Feizi, Ten; Soldati-Favre, Dominique; Matthews, Stephen; Macaire, Héloïse; Riquet, Aurélien; Moncollin, Vincent; Biémont-Trescol, Marie-Claude; Duc Dodon, Madeleine; Hermine, Olivier; Debaud, Anne-Laure; Mahieux, Renaud; Mesnard, Jean-Michel; Pierre, Marlène; Gazzolo, Louis; Bonnefoy, Nathalie; Valentin, Hélène