日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

When Metal Complexes Evolve, and a Minor Species is the Most Active: the Case of Bis(Phenanthroline)Copper in the Catalysis of Glutathione Oxidation and Hydroxyl Radical Generation

当金属络合物演化时,一种次要物种活性最高:以双(菲咯啉)铜催化谷胱甘肽氧化和羟基自由基生成为例

Falcone, Enrico; Vigna, Vincenzo; Schueffl, Hemma; Stellato, Francesco; Vileno, Bertrand; Bouraguba, Merwan; Mazzone, Gloria; Proux, Olivier; Morante, Silvia; Heffeter, Petra; Sicilia, Emilia; Faller, Peter

The anticancer thiosemicarbazone triapine exerts immune-enhancing activities via immunogenic cell death induction and FAS upregulation

抗癌硫代氨基脲三嗪类化合物通过诱导免疫原性细胞死亡和上调FAS发挥免疫增强作用。

Stiller, Bianca; Stefanelli, Alessia; Schueffl, Hemma; Mathuber, Marlene; Skorokhyd, Nadiya; Gufler, Judith; Pirker, Christine; Holcmann, Martin; Panchuk, Rostyslav; Sibilia, Maria; Marko, Doris; Berger, Walter; Kowol, Christian R; Hager, Sonja; Heffeter, Petra

Site-Selectively Functionalized Albumin with DFO*Maleimide for (89)Zr-Radiolabeling Yields a Metabolically Stable PET Probe that Enables Late Time-Point Tumor Imaging in Mice.

用 DFO*马来酰亚胺对白蛋白进行位点选择性功能化,用于 (89)Zr 放射性标记,可产生代谢稳定的 PET 探针,从而实现小鼠的晚期肿瘤成像

Kronberger Julia, Balber Theresa, Schueffl Hemma, Wahrmann Raphaela, Federa Anja, Gradl Mathias, Brandt Marie R, Wanek Thomas, Mitterhauser Markus, Kowol Christian R, Mindt Thomas L, Heffeter Petra

A new fluorescent oxaliplatin(iv) complex with EGFR-inhibiting properties for the treatment of drug-resistant cancer cells

一种新型荧光奥沙利铂(IV)复合物,具有EGFR抑制特性,可用于治疗耐药癌细胞。

Caban, Monika; Fronik, Philipp; Terenzi, Alessio; Federa, Anja; Bormio Nunes, Julia H; Pitek, Rastislav; Kirchhofer, Dominik; Schueffl, Hemma H; Berger, Walter; Keppler, Bernhard K; Kowol, Christian R; Heffeter, Petra

Exploring the Structure-Activity Relationships of Albumin-Targeted Picoplatin-Based Platinum(IV) Prodrugs

探索以白蛋白为靶点的吡啶铂基铂(IV)前药的构效关系

Dijkstra, Martijn; Schueffl, Hemma; Adamova, Barbora; Baumfried, Oliver; Kastner, Alexander; Berger, Walter; Keppler, Bernhard K; Heffeter, Petra; Kowol, Christian R

Novel Maleimide Linkers Based on a Piperazine Motif for Strongly Increased Aqueous Solubility

基于哌嗪基团的新型马来酰亚胺连接剂可显著提高水溶性

Dijkstra, Martijn; Schueffl, Hemma; Federa, Anja; Kast, Caroline; Unterlercher, Alexander; Keppler, Bernhard K; Heffeter, Petra; Kowol, Christian R

Comparative Evaluation of Thiol- and Amine-Conjugating Moieties for Endogenous Albumin Binding after Intravenous Administration.

静脉注射后硫醇和胺结合部分与内源性白蛋白结合的比较评价

Federa Anja, Schueffl Hemma, Minichmayr Iris K, Kastner Alexander, Kronberger Julia, Mindt Thomas L, Heffeter Petra, Kowol Christian R

Insertion of (Bioactive) Equatorial Ligands into Platinum(IV) Complexes

将(生物活性)赤道配体插入铂(IV)配合物中

Kastner, Alexander; Schueffl, Hemma; Yassemipour, Patrick A; Keppler, Bernhard K; Heffeter, Petra; Kowol, Christian R

Einbau von (Bioaktiven) Äquatorialen Liganden in Platin(IV)-Komplexe

将(生物活性)赤道配体引入铂(IV)配合物中

Kastner, Alexander; Schueffl, Hemma; Yassemipour, Patrick A; Keppler, Bernhard K; Heffeter, Petra; Kowol, Christian R