日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Potent and Selective MTH1 Inhibitors for Oncology: Enabling Rapid Target (In)Validation

发现用于肿瘤治疗的高效选择性MTH1抑制剂:实现靶点(不)验证的快速开展

Farand, Julie; Kropf, Jeffrey E; Blomgren, Peter; Xu, Jianjun; Schmitt, Aaron C; Newby, Zachary E; Wang, Ting; Murakami, Eisuke; Barauskas, Ona; Sudhamsu, Jawahar; Feng, Joy Y; Niedziela-Majka, Anita; Schultz, Brian E; Schwartz, Karen; Viatchenko-Karpinski, Serge; Kornyeyev, Dmytro; Kashishian, Adam; Fan, Peidong; Chen, Xiaowu; Lansdon, Eric B; Ports, Michael O; Currie, Kevin S; Watkins, William J; Notte, Gregory T

Biochemical characterization of recombinant influenza A polymerase heterotrimer complex: Polymerase activity and mechanisms of action of nucleotide analogs

重组甲型流感病毒聚合酶异源三聚体复合物的生化特性:聚合酶活性和核苷酸类似物的作用机制

Barauskas, Ona; Xing, Weimei; Aguayo, Esmeralda; Willkom, Madeleine; Sapre, Annapurna; Clarke, Michael; Birkus, Gabriel; Schultz, Brian E; Sakowicz, Roman; Kwon, HyockJoo; Feng, Joy Y

Biochemical characterization of recombinant influenza A polymerase heterotrimer complex: Endonuclease activity and evaluation of inhibitors.

重组甲型流感聚合酶异三聚体复合物的生化特性:核酸内切酶活性及抑制剂评价

Xing Weimei, Barauskas Ona, Kirschberg Thorsten, Niedziela-Majka Anita, Clarke Michael, Birkus Gabriel, Weissburg Perry, Liu Xiaohong, Schultz Brian E, Sakowicz Roman, Kwon HyockJoo, Feng Joy Y