日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

SuFEx-based antitubercular compound irreversibly inhibits Pks13

基于 SuFEx 的抗结核化合物不可逆地抑制 Pks13

Krieger, Inna V; Sukheja, Paridhi; Yang, Baiyuan; Tang, Su; Selle, Daniel; Woods, Ashley; Engelhart, Curtis; Kumar, Pradeep; Harbut, Michael B; Liu, Dongdong; Tsuda, Brendan; Qin, Bo; Bare, Grant A L; Li, Gencheng; Chi, Victor; Gambacurta, Julian; Hvizdos, Janine; Reagan, Matthew; Jones, Isabelle L; Massoudi, Lisa M; Woolhiser, Lisa K; Cascioferro, Alessandro; Kundrick, Erica; Singh, Parul; Reiley, William; Ioerger, Thomas R; Kandula, Dilipkumar Reddy; McCabe, Jacob W; Guo, Taijie; Alland, David; Boshoff, Helena I; Schnappinger, Dirk; Robertson, Gregory T; Mdluli, Khisi; Lee, Kyoung-Jin; Dong, Jiajia; Li, Shuangwei; Schultz, Peter G; Joseph, Sean B; Love, Melissa S; Sharpless, K Barry; Petrassi, H Michael; Chatterjee, Arnab K; Sacchettini, James C; McNamara, Case W

A chemical epigenetic tool to probe site-specific DNA-binding protein complexes

一种用于探测位点特异性DNA结合蛋白复合物的化学表观遗传学工具

Zhu, Jiajun; Li, Zhucui; Xue, Dongxiang; Meng, Zihe; Shao, Sida; Pulecio, Julian; Zhang, Guoan; Huangfu, Danwei; Evans, Todd; Chen, Shuibing; Schultz, Peter G

Targeted degradation of α-Synuclein using an evolved botulinum toxin protease

利用进化的肉毒杆菌毒素蛋白酶靶向降解α-突触核蛋白

Sondermann, Philipp; Diercks, Christian S; Rong, Cynthia; Schultz, Peter G

Targeted protein degradation by KLHDC2 ligands identified by high-throughput screening.

通过高通量筛选鉴定出KLHDC2配体对蛋白质的靶向降解作用

Zhou Han, Zhou Tonglian, Yu Wenli, Liu Liping, Ko Yeonjin, Johnson Kristen A, Wilson Ian A, Schultz Peter G, Bollong Michael J

Targeted Protein Degradation by KLHDC2 Ligands Identified by High Throughput Screening

高通量筛选鉴定出KLHDC2配体靶向降解蛋白质

Zhou, Han; Zhou, Tongliang; Yu, Wenli; Liu, Liping; Ko, Yeonjin; Johnson, Kristen A; Wilson, Ian A; Schultz, Peter G; Bollong, Michael J

A Chemical Epigenetic Probe to Capture the Site-Specific DNA-Binding Protein Complex.

一种用于捕获位点特异性DNA结合蛋白复合物的化学表观遗传探针

Zhu Jiajun, Li Zhucui, Xue Dongxiang, Meng Zihe, Shao Sida, Pulecio Julian, Zhang Guoan, Huangfu Danwei, Evans Todd, Schultz Peter G, Chen Shuibing

Synthesis at the Interface of Chemistry and Biology

化学与生物学交叉领域的合成

Schultz, Peter G

Discovery of CMX990: A Potent SARS-CoV-2 3CL Protease Inhibitor Bearing a Novel Warhead

CMX990 的发现:一种带有新型弹头的强效 SARS-CoV-2 3CL 蛋白酶抑制剂

Dayan Elshan, N G R; Wolff, Karen C; Riva, Laura; Woods, Ashley K; Grabovyi, Gennadii; Wilson, Katy; Pedroarena, James; Ghorai, Sourav; Nazarian, Armen; Weiss, Frank; Liu, Yuyin; Mazumdar, Wrickban; Song, Lirui; Okwor, Neechi; Malvin, Jacqueline; Bakowski, Malina A; Beutler, Nathan; Kirkpatrick, Melanie G; Gebara-Lamb, Amal; Huang, Edward; Nguyen-Tran, Vân T B; Chi, Victor; Li, Shuangwei; Rogers, Thomas F; McNamara, Case W; Gupta, Anil Kumar; Rahimi, Alireza; Chen, Jian Jeffrey; Joseph, Sean B; Schultz, Peter G; Chatterjee, Arnab K

Correction to "Discovery of CMX990: A Potent SARS-CoV-2 3CL Protease Inhibitor Bearing a Novel Warhead"

对“CMX990的发现:一种带有新型弹头的强效SARS-CoV-2 3CL蛋白酶抑制剂”一文的更正

Elshan, N G R Dayan; Wolff, Karen C; Riva, Laura; Woods, Ashley K; Grabovyi, Gennadii; Wilson, Katy; Pedroarena, James; Ghorai, Sourav; Nazarian, Armen; Weiss, Frank; Liu, Yuyin; Mazumdar, Wrickban; Song, Lirui; Okwor, Neechi; Malvin, Jacqueline; Liu, Dongdong; Bakowski, Malina A; Beutler, Nathan; Kirkpatrick, Melanie G; Gebara-Lamb, Amal; Huang, Edward; Nguyen-Tran, Vân T B; Chi, Victor; Li, Shuangwei; Rogers, Thomas F; McNamara, Case W; Gupta, Anil Kumar; Rahimi, Alireza; Chen, Jian Jeffrey; Joseph, Sean B; Schultz, Peter G; Chatterjee, Arnab K

Recent advances in the expanding genetic code

基因组扩展技术的最新进展

Pigula, Michael L; Schultz, Peter G