日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Advances in BRET probes for intracellular target engagement studies

用于细胞内靶标结合研究的BRET探针的进展

Capener, Jacob L; Schwalm, Martin P; Vasta, James D; Michaud, Ani; Teske, Kelly A; Marsiglia, William M; Huber, Kilian V M; Dar, Arvin C; Knapp, Stefan; Axtman, Alison D; Robers, Matthew B

Biochemical investigation of LC3/GABARAP-ligand interaction as an important quality measure for LC3/GABARAP-targeting small molecules: addendum to the guidelines (4th edition)

LC3/GABARAP-配体相互作用的生化研究作为LC3/GABARAP靶向小分子药物的重要质量指标:指南补充(第四版)

Schwalm, Martin P; Lenz, Christopher; Saxena, Krishna; Klionsky, Daniel J; Proschak, Ewgenij; Knapp, Stefan

Cysteine-reactive covalent chloro-N-acetamide ligands induce ferroptosis mediated cell death.

半胱氨酸反应性共价氯-N-乙酰胺配体诱导铁死亡介导的细胞死亡。

Gotthardt Gina, Weckesser Janik, Tascher Georg, Barros da Gama Sara, Uckelmann Hannah J, Sun Shibo, Schwalm Martin P, Mosler Thorsten, Ferrario Giulio, Friedmann Angeli José Pedro, Münch Christian, Knapp Stefan, Müller Stefan

Crystallographic fragment screening reveals ligand hotspots in TRIM21 PRY-SPRY domain.

晶体学片段筛选揭示了TRIM21 PRY-SPRY结构域中的配体热点

Kim Yeojin, Lučić Aleksandar, Lenz Christopher, Farges Frederic, Schwalm Martin P, Saxena Krishna, Hanke Thomas, Marples Peter G, Aschenbrenner Jasmin C, Fearon Daren, von Delft Frank, Krämer Andreas, Knapp Stefan

Inhibition of DYRK1B BY C81 impedes inflammatory processes in leukocytes by reducing STAT3 activity.

C81 通过抑制 DYRK1B 来降低 STAT3 活性,从而阻碍白细胞中的炎症过程

Ciurus Sarah, Elewa Mohammed A F, Palmer Megan A, Wolf Anne, Hector Mandy, Fuhrmann Dominik C, Thomas Dominique, Gurke Robert, Schwalm Martin P, Berger Lena, Zech Thomas J, Burgers Luisa D, Marschalek Rolf, Geisslinger Gerd, Knapp Stefan, Langmann Thomas, Bracher Franz, Weigert Andreas, Fürst Robert

Workflow for E3 Ligase Ligand Validation for PROTAC Development

PROTAC 开发中 E3 连接酶配体验证的工作流程

Miletić, Nebojša; Weckesser, Janik; Mosler, Thorsten; Rathore, Rajeshwari; Hoffmann, Marina E; Gehrtz, Paul; Schlesiger, Sarah; Hartung, Ingo V; Berner, Nicola; Wilhelm, Stephanie; Müller, Juliane; Adhikari, Bikash; Němec, Václav; Sivashanmugam, Saran Aswathaman; Elson, Lewis; Holzmann, Hanna; Schwalm, Martin P; Hoffmann, Lasse; Abdul Azeez, Kamal Rayees; Müller, Susanne; Kuster, Bernhard; Wolf, Elmar; Đikić, Ivan; Knapp, Stefan

Functional Characterization of Pathway Inhibitors for the Ubiquitin-Proteasome System (UPS) as Tool Compounds for CRBN and VHL-Mediated Targeted Protein Degradation.

泛素-蛋白酶体系统 (UPS) 通路抑制剂的功能表征,作为 CRBN 和 VHL 介导的靶向蛋白质降解的工具化合物

Schwalm Martin P, Menge Amelie, Elson Lewis, Greco Francesco A, Robers Matthew B, Müller Susanne, Knapp Stefan

tracerDB: a crowdsourced fluorescent tracer database for target engagement analysis

tracerDB:一个用于靶标结合分析的众包荧光示踪剂数据库

Dopfer, Johannes; Vasta, James D; Müller, Susanne; Knapp, Stefan; Robers, Matthew B; Schwalm, Martin P