日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Click. Screen. Degrade. A Miniaturized D2B Workflow for Rapid PROTAC Discovery

点击。屏幕。降级。用于快速 PROTAC 发现的微型化 D2B 工作流程

Mitrović, Marko; Greco, Francesco Aleksy; García, Yiliam Cruz; Lučić, Aleksandar; Hoffmann, Lasse; Chander, Rohit; Schönfeld, Julia; Liebisch, Nick; Sivashanmugam, Saran Aswathaman; Schwalm, Martin Peter; Egner, Markus; Lewandowski, Max; Merk, Daniel; Morasch, Viktoria; Wolf, Elmar; Müller, Susanne; Hanke, Thomas; Proschak, Ewgenij; Hiesinger, Kerstin; Knapp, Stefan

Un-LOK-ing a New Approach for Conformational Selective Targeting of STK10 (LOK)

针对 STK10 (LOK) 构象选择性靶向的新方法——解构 LOK

Dettenhöfer, Martina; Tandara, Laura Nadine; Amrhein, Jennifer Alisa; Kurz, Christian Georg; Schwalm, Martin Peter; Mensing, Theresa Elisabeth; Wahl, Laurenz Maximilian; Krämer, Andreas; Gerninghaus, Joshua; Lenz, Christopher; Elson, Lewis; Berger, Benedict-Tilman; Schröder, Martin; Saxena, Krishna; Müller, Susanne; Knapp, Stefan; Greco, Francesco Aleksy; Hanke, Thomas

Repurposing of the RIPK1-Selective Benzo[1,4]oxazepin-4-one Scaffold for the Development of a Type III LIMK1/2 Inhibitor.

RIPK1 选择性苯并[1,4]氧氮杂环庚酮-4-酮骨架的再利用,用于开发 III 型 LIMK1/2 抑制剂

Mandel Sebastian, Hanke Thomas, Mathea Sebastian, Chatterjee Deep, Saraswati Hayuningbudi, Berger Benedict-Tilman, Schwalm Martin Peter, Yamamoto Satoshi, Tawada Michiko, Takagi Terufumi, Ahmed Mahmood, Röhm Sandra, Corrionero Ana, Alfonso Patricia, Baena Maria, Elson Lewis, Menge Amelie, Krämer Andreas, Pereira Raquel, Müller Susanne, Krause Daniela S, Knapp Stefan

Discovery of an exquisitely selective WDR5 chemical probe accelerated by a high-quality DEL-ML Hit

高质量的DEL-ML命中加速了极具选择性的WDR5化学探针的发现

Hoffmann, Lasse; Lenz, Christopher; Farges, Frederic; Kimani, Serah W; Dopfer, Johannes; Keller, Sabrina; Schwalm, Martin Peter; Holzmann, Hanna; Kraemer, Andreas; Dong, Aiping; Li, Fengling; Chau, Irene; Halabelian, Levon; Gstaiger, Matthias; Müller, Susanne; Knapp, Stefan; Němec, Václav