日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Nucleobase catalysts for the enzymatic activation of 8-oxoguanine DNA glycosylase 1

核碱基催化剂用于8-氧鸟嘌呤DNA糖基化酶1的酶促活化

Hank, Emily C; D'Arcy-Evans, Nicholas D; Scaletti, Emma Rose; Benítez-Buelga, Carlos; Wallner, Olov; Ortis, Florian; Zhou, Kaixin; Meng, Liuzhen; Del Prado, Alicia; Calvo, Patricia; Almlöf, Ingrid; Wiita, Elisée; Nierlin, Karen; Košenina, Sara; Krämer, Andreas; Eddershaw, Alice; Kehler, Mario; Long, Maeve; Jemth, Ann-Sofie; Dawson, Holly; Stewart, Josephine; Dickey, Adam; Astorga, Mikhael E; Varga, Marek; Homan, Evert J; Scobie, Martin; Knapp, Stefan; Sastre, Leandro; Stenmark, Pål; de Vega, Miguel; Helleday, Thomas; Michel, Maurice

Virtual fragment screening for DNA repair inhibitors in vast chemical space.

在广阔的化学空间中对DNA修复抑制剂进行虚拟片段筛选

Luttens Andreas, Vo Duc Duy, Scaletti Emma R, Wiita Elisée, Almlöf Ingrid, Wallner Olov, Davies Jonathan, Košenina Sara, Meng Liuzhen, Long Maeve, Mortusewicz Oliver, Masuyer Geoffrey, Ballante Flavio, Michel Maurice, Homan Evert, Scobie Martin, Kalderén Christina, Warpman Berglund Ulrika, Tarnovskiy Andrii V, Radchenko Dmytro S, Moroz Yurii S, Kihlberg Jan, Stenmark Pål, Helleday Thomas, Carlsson Jens

Giving an Enzyme Scissors: Serotonin Derivatives as Potent Organocatalytic Switches for DNA Repair Enzyme OGG1

赋予酶剪刀:血清素衍生物作为DNA修复酶OGG1的强效有机催化开关

Varga, Marek; Ortis, Florian; Del Prado, Alicia; Eddershaw, Alice; Scaletti Hutchinson, Emma; Hank, Emily C; Zhou, Kaixin; Rudolfová, Natálie; Dodaro, Alessia; Wiita, Elisée; Almlöf, Ingrid; Karsten, Stella; Mamonov, Kirill; Ahmed, Sara H; Bentley, Kirsty; Wallner, Olov; Homan, Evert J; Scobie, Martin; Helleday, Thomas; Prejanò, Mario; Stenmark, Pål; de Vega, Miguel; Watson, Allan J B; Michel, Maurice

Topical MTH1 Inhibition Suppresses SKP2-WNT5a-Driven Psoriatic Hyperproliferation

局部应用MTH1抑制剂可抑制SKP2-WNT5a驱动的银屑病细胞过度增殖。

Bivik Eding, Cecilia; Köhler, Ines; Moparthi, Lavanya; Sjögren, Florence; Andersson, Blanka; Das, Debojyoti; Verma, Deepti; Scobie, Martin; Warpman Berglund, Ulrika; Enerbäck, Charlotta

The anabolic steroid stanozolol is a potent inhibitor of human MutT homolog 1

合成代谢类固醇司坦唑醇是人类 MutT 同源物 1 的强效抑制剂。

Scaletti Hutchinson, Emma; Gustafsson Westergren, Robert; Almlöf, Ingrid; Jemth, Ann-Sofie; Scobie, Martin; Warpman Berglund, Ulrika; Helleday, Thomas; Stenmark, Pål

Crystal structures of NUDT15 variants enabled by a potent inhibitor reveal the structural basis for thiopurine sensitivity

利用强效抑制剂解析的NUDT15变体晶体结构揭示了硫嘌呤敏感性的结构基础。

Rehling, Daniel; Zhang, Si Min; Jemth, Ann-Sofie; Koolmeister, Tobias; Throup, Adam; Wallner, Olov; Scaletti, Emma; Moriyama, Takaya; Nishii, Rina; Davies, Jonathan; Desroses, Matthieu; Rudd, Sean G; Scobie, Martin; Homan, Evert; Berglund, Ulrika Warpman; Yang, Jun J; Helleday, Thomas; Stenmark, Pål

Correction: A patient-derived xenograft pre-clinical trial reveals treatment responses and a resistance mechanism to karonudib in metastatic melanoma

更正:一项患者来源的异种移植临床前试验揭示了转移性黑色素瘤对卡罗努迪布的治疗反应和耐药机制

Einarsdottir, Berglind O; Karlsson, Joakim; Söderberg, Elin M V; Lindberg, Mattias F; Funck-Brentano, Elisa; Jespersen, Henrik; Brynjolfsson, Siggeir F; Bagge, Roger Olofsson; Carstam, Louise; Scobie, Martin; Koolmeister, Tobias; Wallner, Olof; Stierner, Ulrika; Berglund, Ulrika Warpman; Ny, Lars; Nilsson, Lisa M; Larsson, Erik; Helleday, Thomas; Nilsson, Jonas A

Structure-metabolism-relationships in the microsomal clearance of piperazin-1-ylpyridazines

哌嗪-1-基哒嗪微粒体清除的结构-代谢关系

Llona-Minguez, Sabin; Ghassemian, Artin; Baranczewski, Pawel; Desroses, Matthieu; Koolmeister, Tobias; Artursson, Per; Scobie, Martin; Helleday, Thomas

Discovery of the First Potent and Selective Inhibitors of Human dCTP Pyrophosphatase 1

人类 dCTP 焦磷酸酶 1 的首个高效选择性抑制剂的发现

Llona-Minguez, Sabin; Höglund, Andreas; Jacques, Sylvain A; Johansson, Lars; Calderón-Montaño, José Manuel; Claesson, Magnus; Loseva, Olga; Valerie, Nicholas C K; Lundbäck, Thomas; Piedrafita, Javier; Maga, Giovanni; Crespan, Emmanuele; Meijer, Laurent; Morón, Estefanía Burgos; Baranczewski, Pawel; Hagbjörk, Ann-Louise; Svensson, Richard; Wiita, Elisee; Almlöf, Ingrid; Visnes, Torkild; Jeppsson, Fredrik; Sigmundsson, Kristmundur; Jensen, Annika Jenmalm; Artursson, Per; Jemth, Ann-Sofie; Stenmark, Pål; Berglund, Ulrika Warpman; Scobie, Martin; Helleday, Thomas