日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Novel Proline-Based Neuropeptide FF Receptor Antagonists

发现新型脯氨酸类神经肽 FF 受体拮抗剂

Thuy Nguyen, Ann M Decker, Tiffany L Langston, Kelly M Mathews, Justin N Siemian, Jun-Xu Li, Danni L Harris, Scott P Runyon, Yanan Zhang

Identification of N-[(5-{[(4-methylphenyl)sulfonyl]amino}-3-(trifluoroacetyl)-1H-indol-1-yl)acetyl]-l-leucine (NTRC-824), a neurotensin-like nonpeptide compound selective for the neurotensin receptor type 2

鉴定 N-[(5-{[(4-甲基苯基)磺酰基]氨基}-3-(三氟乙酰基)-1H-吲哚-1-基)乙酰基]-l-亮氨酸 (NTRC-824),一种选择性作用于 2 型神经降压素受体的神经降压素样非肽化合物

James B Thomas, Angela M Giddings, Robert W Wiethe, Srinivas Olepu, Keith R Warner, Philippe Sarret, Louis Gendron, Jean-Michel Longpre, Yanan Zhang, Scott P Runyon, Brian P Gilmour

Enhanced bioactivity of silybin B methylation products

水飞蓟宾 B 甲基化产物的增强生物活性

Arlene A Sy-Cordero, Tyler N Graf, Scott P Runyon, Mansukh C Wani, David J Kroll, Rajesh Agarwal, Scott J Brantley, Mary F Paine, Stephen J Polyak, Nicholas H Oberlies