日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of spirodioxolane nsP2 helicase inhibitors with antialphaviral activity

鉴定具有抗甲病毒活性的螺二氧戊环nsP2解旋酶抑制剂

Oh, Hans J; Sears, John D; Ramalingam, Bose Muthu; Saleem, Rahman Shah Zaib; Davis-Gilbert, Zachary W; Hossain, Mohammed Anwar; Moorman, Stella R; Ohja, Durbadal; Martinez, Sabian A; Burdick, Jane E; Couñago, Rafael M; Moorman, Nathaniel J; Heise, Mark T; Todd, Matthew H; Willson, Timothy M

RNA-targeted proteomics identifies YBX1 as critical for efficient HCMV mRNA translation.

RNA靶向蛋白质组学鉴定出YBX1对于HCMV mRNA的有效翻译至关重要

Dickmander Rebekah J, Lenarcic Erik M, Sears John D, Hale Andrew E, Moorman Nathaniel J

Identification of Direct-Acting nsP2 Helicase Inhibitors with Antialphaviral Activity

鉴定具有抗甲病毒活性的直接作用nsP2解旋酶抑制剂

Muthu Ramalingam, Bose; Sears, John D; Talbot, Kacey M; Su, Yuan-Wei Norman; Houliston, Scott; Hossain, Mohammed Anwar; Davis-Gilbert, Zachary W; Zhao, Chunqing; Oh, Hans J; Brown, Peter J; Sanders, Marcia K; Moorman, Stella R; Ojha, Durbadal; Burdick, Jane E; Law, Isabella; Morales, Noah L; Martinez, Sabian A; Loppnau, Peter; Garcia Perez, Julia; Drobish, Adam M; Morrison, Thomas E; Streblow, Zachary J; Streblow, Daniel N; Arrowsmith, Cheryl H; Vargason, Ava; Couñago, Rafael M; Halabelian, Levon; Arnold, Jamie J; Cameron, Craig E; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

N-Alkyl Sulfamates as a New Class of nsP2 Cysteine Protease Inhibitors with Broad-Spectrum Antialphaviral Activity

N-烷基氨基磺酸酯作为一类新型nsP2半胱氨酸蛋白酶抑制剂,具有广谱抗甲病毒活性

Ghoshal, Anirban; Sears, John D; Hossain, Mohammad Anwar; Tse, Edwin G; Howell, Stefanie; Burdick, Jane E; Morales, Noah L; Martinez, Sabian A; Law, Isabella; Streblow, Zachary J; Streblow, Daniel N; Couñago, Rafael M; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

Enantioselective Chemical Probe for Chikungunya nsP2 Helicase with Antialphaviral Activity

具有抗甲病毒活性的基孔肯雅病毒nsP2解旋酶对映选择性化学探针

Muthu Ramalingam, Bose; Oh, Hans J; Sears, John D; Chen, Chun-Hsing; Vala, Anand; Liu, Shubin; Talbot, Kacey M; Hossain, Mohammed Anwar; Brown, Peter J; Houliston, Scott; Garcia Perez, Julia; Li, Fengling; Amare, Meareg G; Halfmann, Peter; Smith, Jessica L; Hirsch, Alec J; Arrowsmith, Cheryl H; Halabelian, Levon; Vargason, Ava; Couñago, Rafael M; Arnold, Jamie J; Cameron, Craig E; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

Novel Computational Pipeline to Identify Target Sites for Broad Spectrum Antiviral Drugs

用于识别广谱抗病毒药物靶点的新型计算流程

Sears, John D; Popov, Konstantin I; Sylvester, Paul; Dickmander, Rebekah; Loome-Diaz, Jennifer; Chang, Che-Kang; Huff, Julia; Sanders, Wes; Saba, Nicholas A; Sorensen, Madeleine; Drobish, Adam M; May, Nicholas A; Namitz, Kevin; Fecko, Julia; Arnold, Jamie J; Yennawar, Neela H; Cameron, Craig E; Morrison, Thomas E; Tropsha, Alexander; Heise, Mark T; Moorman, Nathaniel J

Identification of a cell-active chikungunya virus nsP2 protease inhibitor using a covalent fragment-based screening approach

利用共价片段筛选方法鉴定具有细胞活性的基孔肯雅病毒nsP2蛋白酶抑制剂

Merten, Eric M; Sears, John D; Leisner, Tina M; Hardy, P Brian; Ghoshal, Anirban; Hossain, Mohammad Anwar; Asressu, Kesatebrhan Haile; Brown, Peter J; Tse, Edwin G; Stashko, Michael A; Li, Kelin; Norris-Drouin, Jacqueline L; Herring, Laura E; Mordant, Angie L; Webb, Thomas S; Mills, Christine A; Barker, Natalie K; Streblow, Zachary J; Perveen, Sumera; Arrowsmith, Cheryl H; Couñago, Rafael Miguez; Arnold, Jamie J; Cameron, Craig E; Streblow, Daniel N; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M; Popov, Konstantin I; Pearce, Kenneth H

Structure Activity of β-Amidomethyl Vinyl Sulfones as Covalent Inhibitors of Chikungunya nsP2 Cysteine Protease with Antialphavirus Activity

β-酰胺甲基乙烯基砜作为基孔肯雅病毒nsP2半胱氨酸蛋白酶共价抑制剂的结构活性及其抗甲病毒活性

Ghoshal, Anirban; Asressu, Kesatebrhan Haile; Hossain, Mohammad Anwar; Brown, Peter J; Nandakumar, Meganathan; Vala, Anand; Merten, Eric M; Sears, John D; Law, Isabella; Burdick, Jane E; Morales, Noah L; Perveen, Sumera; Pearce, Kenneth H; Popov, Konstantin I; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

Transcriptome analysis reveals organ-specific effects of 2-deoxyglucose treatment in healthy mice

转录组分析揭示了2-脱氧葡萄糖治疗对健康小鼠器官的特异性影响

Wells, Ann E; Wilson, John J; Heuer, Sarah E; Sears, John D; Wei, Jian; Pandey, Raghav; Costa, Mauro W; Kaczorowski, Catherine C; Roopenian, Derry C; Chang, Chih-Hao; Carter, Gregory W

Structure Activity of β-Amidomethyl Vinyl Sulfones as Covalent Inhibitors of Chikungunya nsP2 Cysteine Protease with Anti-alphavirus Activity

β-酰胺甲基乙烯基砜作为基孔肯雅病毒nsP2半胱氨酸蛋白酶共价抑制剂的结构活性及其抗甲病毒活性

Ghoshal, Anirban; Asressu, Kesatebrhan Haile; Hossain, Mohammad Anwar; Brown, Peter J; Merten, Eric M; Sears, John D; Perveen, Sumera; Pearce, Kenneth H; Popov, Konstantin I; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M