Structure-Guided Design of a KMT9 Inhibitor Prodrug with Cellular Activity.
基于结构的KMT9抑制剂前药设计及其细胞活性
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c02953
Wang Sheng, Barthes Nicolas P F, Urban Sylvia, Hazai Viktor I, Klein Sebastian O, Pappert Tabea, Kümmel Paul, Heller Nicolas, Bacher Johannes, Staudt Maximilian, Ruprecht Jan, Peng Ling, Sum Manuela, Berlin Christopher, Sarraf Daad, Regenass Pierre, Warstat Robin, Walz Johannes, Mishra Pankaj, Zhang Lin, Einsle Oliver, Günther Stefan, Breit Bernhard, Metzger Eric, Jung Manfred, Schüle Roland