Alkyne Two-Phase Strategy: Rapid Generation of TK-285-Derived PROTACs as BRD4 Degraders
炔烃两相策略:快速生成TK-285衍生的PROTACs作为BRD4降解剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c03771
Yamakoshi, Hiroyuki; Watanabe, Ryo; Segawa, Ryosuke; Ishihara, Ryosuke; Tachibana, Ryo; Kudo, Genki; Nagasawa, Shota; Yamanaka, Satoshi; Ito, Ayano; Takeda, Hiroyuki; Sawasaki, Tatsuya; Yoshino, Ryunosuke; Hirokawa, Takatsugu; Doi, Takayuki; Hirasawa, Noriyasu; Iwabuchi, Yoshiharu