日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Venetoclax resistance in preclinical KMT2A-rearranged acute lymphoblastic leukemia models is characterized by high inter- and intra-model heterogeneity

在临床前KMT2A重排急性淋巴细胞白血病模型中,维奈托克耐药性的特征是模型间和模型内异质性较高。

Richter, Anna; Kinsky, Lea; Lange, Sandra; Trakooljul, Nares; Hadlich, Frieder; Sekora, Anett; Knuebel, Gudrun; Krohn, Saskia; Schmidt, Christian; Busch, Michelle; Schreiber, Tim; Kumstel, Simone; Wimmers, Klaus; Murua Escobar, Hugo; Junghanss, Christian

Exploring Thiazolopyridine AV25R: Unraveling of Biological Activities, Selective Anti-Cancer Properties and In Silico Target and Binding Prediction in Hematological Neoplasms

探索噻唑并吡啶类化合物AV25R:揭示其在血液肿瘤中的生物活性、选择性抗癌特性以及计算机靶点和结合预测

Ladwig, Annika; Gupta, Shailendra; Ehlers, Peter; Sekora, Anett; Alammar, Moosheer; Koczan, Dirk; Wolkenhauer, Olaf; Junghanss, Christian; Langer, Peter; Murua Escobar, Hugo

Effective tumor cell abrogation via Venetoclax-mediated BCL-2 inhibition in KMT2A-rearranged acute B-lymphoblastic leukemia

在KMT2A重排的急性B淋巴细胞白血病中,Venetoclax通过BCL-2抑制有效清除肿瘤细胞

Richter, Anna; Lange, Sandra; Holz, Clemens; Brock, Luisa; Freitag, Thomas; Sekora, Anett; Knuebel, Gudrun; Krohn, Saskia; Schwarz, Rico; Hinz, Burkhard; Murua Escobar, Hugo; Junghanss, Christian

Spirooxindol-1,3-oxazine Alkaloids: Highly Potent and Selective Antitumor Agents Evolved from Iterative Structure Optimization

螺环氧吲哚-1,3-噁嗪生物碱:通过迭代结构优化开发的高效选择性抗肿瘤药物

Eichhorst, Annika; Gallhof, Malte; Voss, Alice; Sekora, Anett; Eggers, Leon; Huyen, Le Thi; Junghanss, Christian; Murua Escobar, Hugo; Brasholz, Malte

Combined Application of Pan-AKT Inhibitor MK-2206 and BCL-2 Antagonist Venetoclax in B-Cell Precursor Acute Lymphoblastic Leukemia.

泛AKT抑制剂MK-2206与BCL-2拮抗剂Venetoclax联合应用于B细胞前体急性淋巴细胞白血病

Richter Anna, Fischer Elisabeth, Holz Clemens, Schulze Julia, Lange Sandra, Sekora Anett, Knuebel Gudrun, Henze Larissa, Roolf Catrin, Murua Escobar Hugo, Junghanss Christian

Influence of Casein kinase II inhibitor CX-4945 on BCL6-mediated apoptotic signaling in B-ALL in vitro and in vivo

酪蛋白激酶II抑制剂CX-4945对体外和体内B细胞急性淋巴细胞白血病(B-ALL)中BCL6介导的细胞凋亡信号通路的影响

Richter, Anna; Sender, Sina; Lenz, Annemarie; Schwarz, Rico; Hinz, Burkhard; Knuebel, Gudrun; Sekora, Anett; Murua Escobar, Hugo; Junghanss, Christian; Roolf, Catrin

Novel Isoquinolinamine and Isoindoloquinazolinone Compounds Exhibit Antiproliferative Activity in Acute Lymphoblastic Leukemia Cells

新型异喹啉胺和异吲哚喹唑啉酮化合物对急性淋巴细胞白血病细胞表现出抗增殖活性

Roolf, Catrin; Saleweski, Jan-Niklas; Stein, Arno; Richter, Anna; Maletzki, Claudia; Sekora, Anett; Escobar, Hugo Murua; Wu, Xiao-Feng; Beller, Matthias; Junghanss, Christian

Characterization of the novel indolylmaleimides' PDA-66 and PDA-377 effect on canine lymphoma cells

新型吲哚基马来酰亚胺类化合物PDA-66和PDA-377对犬淋巴瘤细胞作用的特征分析

Liu, Wen; Beck, Julia; Schmidt, Laura C; Roolf, Catrin; Pews-Davtyan, Anahit; Rütgen, Barbara C; Hammer, Sabine; Willenbrock, Saskia; Sekora, Anett; Rolfs, Arndt; Beller, Matthias; Brenig, Bertram; Nolte, Ingo; Junghanss, Christian; Schütz, Ekkehard; Murua Escobar, Hugo

Kinetics of Langerhans cell chimerism in the skin of dogs following 2 Gy TBI allogeneic hematopoietic stem cell transplantation

Gy TBI 同种异体造血干细胞移植后犬皮肤中朗格汉斯细胞嵌合体的动力学

Peters, Sabrina; Junghanss, Christian; Knueppel, Anne; Murua Escobar, Hugo; Roolf, Catrin; Knuebel, Gudrun; Sekora, Anett; Lindner, Iris; Jonas, Ludwig; Freund, Mathias; Lange, Sandra

Polymorphisms of the murine mitochondrial ND4, CYTB and COX3 genes impact hematopoiesis during aging

小鼠线粒体ND4、CYTB和COX3基因的多态性影响衰老过程中的造血作用

Kretzschmar, Christin; Roolf, Catrin; Timmer, Katrin; Sekora, Anett; Knübel, Gudrun; Murua Escobar, Hugo; Fuellen, Georg; Ibrahim, Saleh M; Tiedge, Markus; Baltrusch, Simone; Jaster, Robert; Köhling, Rüdiger; Junghanss, Christian