日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Multiple intramolecular triggers converge to preferential G protein coupling in the CB(2)R

多种分子内触发因素汇聚于CB(2)受体中G蛋白的优先偶联。

Morales-Pastor, Adrian; Miljuš, Tamara; Dieguez-Eceolaza, Miguel; Stępniewski, Tomasz Maciej; Ledesma-Martin, Vicente; Heydenreich, Franziska M; Flock, Tilman; Plouffe, Bianca; Le Gouill, Christian; Duchaine, Jean; Sykes, David A; Nicholson, Colin; Koers, Eline J; Guba, Wolfgang; Rufer, Arne C; Grether, Uwe; Bouvier, Michel; Veprintsev, Dmitry B; Selent, Jana

Large scale investigation of GPCR molecular dynamics data uncovers allosteric sites and lateral gateways

对GPCR分子动力学数据的大规模研究揭示了变构位点和侧向通道

Aranda-García, David; Stepniewski, Tomasz Maciej; Torrens-Fontanals, Mariona; García-Recio, Adrian; Lopez-Balastegui, Marta; Medel-Lacruz, Brian; Morales-Pastor, Adrián; Peralta-García, Alejandro; Dieguez-Eceolaza, Miguel; Sotillo-Nuñez, David; Ding, Tianyi; Drabek, Matthäus; Jacquemard, Célien; Jakowiecki, Jakub; Jespers, Willem; Jiménez-Rosés, Mireia; Jun-Yu-Lim, Víctor; Nicoli, Alessandro; Orzel, Urszula; Shahraki, Aida; Tiemann, Johanna K S; Ledesma-Martin, Vicente; Nerín-Fonz, Francho; Suárez-Dou, Sergio; Canal, Oriol; Pándy-Szekeres, Gáspár; Mao, Jiafei; Gloriam, David E; Kellenberger, Esther; Latek, Dorota; Guixà-González, Ramon; Gutiérrez-de-Terán, Hugo; Tikhonova, Irina G; Hildebrand, Peter W; Filizola, Marta; Babu, M Madan; Di Pizio, Antonella; Filipek, Slawomir; Kolb, Peter; Cordomi, Arnau; Giorgino, Toni; Marti-Solano, Maria; Selent, Jana

An arginine switch drives the stepwise activation of β-arrestin by CXCR7

精氨酸开关驱动 CXCR7 逐步激活 β-arrestin。

Ji, Jeong Seok; Yun, Yaejin; Stepniewski, Tomasz Maciej; Yoon, Hye-Jin; Min, Kyungjin; Park, Ji Young; Chung, Chiwoon; Eceolaza, Miguel Dieguez; Chung, Ka Young; Selent, Jana; Lee, Hyung Ho

Loss-of-function Gα(s) rare disease variants exert mutation-specific effects on GPCR signaling

功能丧失的Gα(s)罕见疾病变异体对GPCR信号传导产生突变特异性影响

Redfern-Nichols, Theo; O'Brien, Shannon L; Huang, Xianglin; Medel-Lacruz, Brian; Calebiro, Davide; Selent, Jana; Ladds, Graham; Marti-Solano, Maria

Type-1 Cannabinoid Receptor Promiscuous Coupling: Computational Insights into Receptor-G Protein Interaction Dynamics

1型大麻素受体混杂偶联:受体-G蛋白相互作用动力学的计算见解

Berghella, Alessandro; Stepniewski, Tomasz Maciej; Sabatucci, Annalaura; Lopez-Balastegui, Marta; Nowicki, Krzysztof; Dufrusine, Beatrice; Selent, Jana; Dainese, Enrico

Computational Design and Evaluation of Peptides to Target SARS-CoV-2 Spike-ACE2 Interaction

利用计算方法设计并评估靶向SARS-CoV-2刺突蛋白-ACE2相互作用的肽段。

Almabhouh, Saja; Cecon, Erika; Basubas, Florence; Molina-Fernandez, Ruben; Maciej Stepniewski, Tomasz; Selent, Jana; Jockers, Ralf; Rahmeh, Amal; Oliva, Baldo; Fernandez-Fuentes, Narcis

Distinctive patterns of G protein coupling induced by the structurally similar 5-HT(2A) receptor ligands ketanserin and altanserin in human prefrontal cortex

结构相似的5-HT(2A)受体配体酮色林和阿坦色林在人类前额叶皮层中诱导的独特G蛋白偶联模式

Miranda-Azpiazu, Patricia; Muguruza, Carolina; Stepniewski, Tomasz Maciej; Muneta-Arrate, Itziar; Moreira, David; Brea, José; Callado, Luis F; Loza, María Isabel; González-Maeso, Javier; Selent, Jana; Diez-Alarcia, Rebeca; Meana, J Javier

Molecular insights into atypical modes of β-arrestin interaction with seven transmembrane receptors

β-arrestin与七次跨膜受体相互作用的非典型模式的分子机制研究

Maharana, Jagannath; Sano, Fumiya K; Sarma, Parishmita; Yadav, Manish K; Duan, Longhan; Stepniewski, Tomasz M; Chaturvedi, Madhu; Ranjan, Ashutosh; Singh, Vinay; Saha, Sayantan; Mahajan, Gargi; Chami, Mohamed; Shihoya, Wataru; Selent, Jana; Chung, Ka Young; Banerjee, Ramanuj; Nureki, Osamu; Shukla, Arun K

AlloViz: A tool for the calculation and visualisation of protein allosteric communication networks

AlloViz:用于计算和可视化蛋白质变构通讯网络的工具

Nerín-Fonz, Francho; Caprai, Camilla; Morales-Pastor, Adrián; Lopez-Balastegui, Marta; Aranda-García, David; Giorgino, Toni; Selent, Jana

SCoV2-MD: a database for the dynamics of the SARS-CoV-2 proteome and variant impact predictions

SCoV2-MD:SARS-CoV-2 蛋白质组动态变化及变异株影响预测数据库

Torrens-Fontanals, Mariona; Peralta-García, Alejandro; Talarico, Carmine; Guixà-González, Ramon; Giorgino, Toni; Selent, Jana