日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Potent and selective SETDB1 covalent negative allosteric modulator reduces methyltransferase activity in cells

强效且选择性的 SETDB1 共价负变构调节剂可降低细胞中的甲基转移酶活性

Mélanie Uguen, Devan J Shell, Madhushika Silva, Yu Deng, Fengling Li, Magdalena M Szewczyk, Ka Yang, Yani Zhao, Michael A Stashko, Jacqueline L Norris-Drouin, Jarod M Waybright, Serap Beldar, Justin M Rectenwald, Angie L Mordant, Thomas S Webb, Laura E Herring, Cheryl H Arrowsmith, Suzanne Ackloo, S

Cdyl Deficiency Brakes Neuronal Excitability and Nociception through Promoting Kcnb1 Transcription in Peripheral Sensory Neurons

Cdyl 缺乏通过促进外周感觉神经元中的 Kcnb1 转录来抑制神经元兴奋性和痛觉

Zhao-Wei Sun, Jarod M Waybright, Serap Beldar, Lu Chen, Caroline A Foley, Jacqueline L Norris-Drouin, Tian-Jie Lyu, Aiping Dong, Jinrong Min, Yu-Pu Wang, Lindsey I James, Yun Wang

PGE1 and PGA1 bind to Nurr1 and activate its transcriptional function

PGE1 和 PGA1 与 Nurr1 结合并激活其转录功能

Sreekanth Rajan #, Yongwoo Jang #, Chun-Hyung Kim #, Woori Kim #, Hui Ting Toh, Jeha Jeon, Bin Song, Aida Serra, Julien Lescar, Jun Yeob Yoo, Serap Beldar, Hong Ye, Congbao Kang, Xue-Wei Liu, Melissa Feitosa, Yeahan Kim, Dabin Hwang, Geraldine Goh, Kah-Leong Lim, Hye Min Park, Choong Hwan Lee, Sungw