日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Multifaceted approach toward mapping out the anticancer properties of small molecules via in vitro evaluation on melanoma and nonmelanoma skin cancer cells, and in silico target fishing

通过对黑色素瘤和非黑色素瘤皮肤癌细胞进行体外评估以及计算机模拟靶向钓鱼,采用多方面方法确定小分子的抗癌特性

Samuel T Boateng, Tithi Roy, Mercy E Agbo, Md Ashiq Mahmud, Sergette Banang-Mbeumi, Roxane-Cherille N Chamcheu, Rajesh K Yadav, Marion Bramwell, Long K Pham, Danny D Dang, Keith E Jackson, Bolni Marius Nagalo, Ronald A Hill, Tatiana Efimova, Jean Fotie, Jean Christopher Chamcheu

Dual targeting of mTOR/IL-17A and autophagy by fisetin alleviates psoriasis-like skin inflammation

漆黄素对 mTOR/IL-17A 和自噬的双重靶向作用可缓解银屑病样皮肤炎症

Tithi Roy, Sergette Banang-Mbeumi, Samuel T Boateng, Emmanuelle M Ruiz, Roxane-Cherille N Chamcheu, Lin Kang, Judy A King, Anthony L Walker, Bolni Marius Nagalo, Konstantin G Kousoulas, Stephane Esnault, Shile Huang, Jean Christopher Chamcheu

Synthesis, in silico modelling, and in vitro biological evaluation of substituted pyrazole derivatives as potential anti-skin cancer, anti-tyrosinase, and antioxidant agents

取代吡唑衍生物作为潜在抗皮肤癌、抗酪氨酸酶和抗氧化剂的合成、计算机模拟和体外生物学评价

Samuel T Boateng, Tithi Roy, Kara Torrey, Uchechi Owunna, Sergette Banang-Mbeumi, David Basnet, Eleonora Niedda, Alexis D Alexander, Denzel El Hage, Siriki Atchimnaidu, Bolni Marius Nagalo, Dinesh Aryal, Ann Findley, Navindra P Seeram, Tatiana Efimova, Mario Sechi, Ronald A Hill, Hang Ma, Jean Chris

The PI3K-Akt-mTOR and Associated Signaling Pathways as Molecular Drivers of Immune-Mediated Inflammatory Skin Diseases: Update on Therapeutic Strategy Using Natural and Synthetic Compounds

PI3K-Akt-mTOR及其相关信号通路作为免疫介导的炎症性皮肤病的分子驱动因素:利用天然和合成化合物的治疗策略最新进展

Roy, Tithi; Boateng, Samuel T; Uddin, Mohammad B; Banang-Mbeumi, Sergette; Yadav, Rajesh K; Bock, Chelsea R; Folahan, Joy T; Siwe-Noundou, Xavier; Walker, Anthony L; King, Judy A; Buerger, Claudia; Huang, Shile; Chamcheu, Jean Christopher

Synthesis, inverse docking-assisted identification and in vitro biological characterization of Flavonol-based analogs of fisetin as c-Kit, CDK2 and mTOR inhibitors against melanoma and non-melanoma skin cancers

合成、逆向对接辅助鉴定和体外生物学表征基于黄酮醇的fisetin类似物作为c-Kit、CDK2和mTOR抑制剂对抗黑色素瘤和非黑色素瘤皮肤癌

Tithi Roy, Samuel T Boateng, Sergette Banang-Mbeumi, Pankaj K Singh, Pratik Basnet, Roxane-Cherille N Chamcheu, Federico Ladu, Isabel Chauvin, Vladimir S Spiegelman, Ronald A Hill, Konstantin G Kousoulas, Bolni Marius Nagalo, Anthony L Walker, Jean Fotie, Siva Murru, Mario Sechi, Jean Christopher Ch

Identification of new fisetin analogs as kinase inhibitors: Data on synthesis and anti-skin cancer activities evaluation

鉴定新型非瑟酮类似物作为激酶抑制剂:合成数据及抗皮肤癌活性评价

Roy, Tithi; Boateng, Samuel T; Banang-Mbeumi, Sergette; Singh, Pankaj K; Basnet, Pratik; Chamcheu, Roxane-Cherille N; Ladu, Federico; Chauvin, Isabel; Spiegelman, Vladimir S; Hill, Ronald A; Kousoulas, Konstantin G; Nagalo, Bolni Marius; Walker, Anthony L; Fotie, Jean; Murru, Siva; Sechi, Mario; Chamcheu, Jean Christopher

Role and Therapeutic Targeting of the PI3K/Akt/mTOR Signaling Pathway in Skin Cancer: A Review of Current Status and Future Trends on Natural and Synthetic Agents Therapy

PI3K/Akt/mTOR信号通路在皮肤癌中的作用及治疗靶点:天然和合成药物治疗现状及未来趋势综述

Chamcheu, Jean Christopher; Roy, Tithi; Uddin, Mohammad Burhan; Banang-Mbeumi, Sergette; Chamcheu, Roxane-Cherille N; Walker, Anthony L; Liu, Yong-Yu; Huang, Shile

Fisetin, a 3,7,3',4'-Tetrahydroxyflavone Inhibits the PI3K/Akt/mTOR and MAPK Pathways and Ameliorates Psoriasis Pathology in 2D and 3D Organotypic Human Inflammatory Skin Models

3,7,3',4'-四羟基黄酮非瑟黄素可抑制 PI3K/Akt/mTOR 和 MAPK 通路,改善 2D 和 3D 器官型人类炎症皮肤模型中的银屑病病理

Jean Christopher Chamcheu, Stephane Esnault, Vaqar M Adhami, Andrea L Noll, Sergette Banang-Mbeumi, Tithi Roy, Sitanshu S Singh, Shile Huang, Konstantin G Kousoulas, Hasan Mukhtar

Graviola (Annona muricata) Exerts Anti-Proliferative, Anti-Clonogenic and Pro-Apoptotic Effects in Human Non-Melanoma Skin Cancer UW-BCC1 and A431 Cells In Vitro: Involvement of Hedgehog Signaling

番荔枝 (Annona muricata) 在体外对人类非黑色素瘤皮肤癌 UW-BCC1 和 A431 细胞发挥抗增殖、抗克隆和促凋亡作用:Hedgehog 信号的参与

Jean Christopher Chamcheu, Islam Rady, Roxane-Cherille N Chamcheu, Abu Bakar Siddique, Melissa B Bloch, Sergette Banang Mbeumi, Abiola S Babatunde, Mohammad B Uddin, Felicite K Noubissi, Peter W Jurutka, Yong-Yu Liu, Vladimir S Spiegelman, G Kerr Whitfield, Khalid A El Sayed

Anticancer Properties of Graviola (Annona muricata): A Comprehensive Mechanistic Review

刺果番荔枝(Annona muricata)的抗癌特性:一项全面的机制综述

Rady, Islam; Bloch, Melissa B; Chamcheu, Roxane-Cherille N; Banang Mbeumi, Sergette; Anwar, Md Rafi; Mohamed, Hadir; Babatunde, Abiola S; Kuiate, Jules-Roger; Noubissi, Felicite K; El Sayed, Khalid A; Whitfield, G Kerr; Chamcheu, Jean Christopher