日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

RNA-binding protein LARP6 coordinates hepatic stellate cell activation and liver fibrosis

RNA结合蛋白LARP6协调肝星状细胞活化和肝纤维化

Kim, Hyun Young; Mizrahi, Orel; Lee, Wonseok; Rosenthal, Sara B; Han, Cuijuan; Yee, Brian A; Blue, Steven M; Diaz, Jesiel; Jonnalagadda, Jyotiprakash P; Street, Lena A; Hokutan, Kanani; Jang, Haeum; Miciano, Charlene; Ma, Chen-Ting; Bobkov, Andrey A; Sergienko, Eduard; Jackson, Michael R; Jovanovic, Marko; Stefanovic, Branko; Kisseleva, Tatiana; Yeo, Gene W; Brenner, David A

Uncompetitive Allosteric Inhibitor of Mitochondrial Creatine Kinase Prevents Binding and Release of Creatine by Stabilization of Loop Closure

线粒体肌酸激酶的非竞争性变构抑制剂通过稳定环路闭合来阻止肌酸的结合和释放。

Demir, Merve; Ma, Chen-Ting; Puvvula, Nikhil; Koepping, Laura; Gosalia, Palak; Pollari, Sirkku; Alba, Shaun; Zong, Zoe; Li, Ya; Fujimoto, Lynn; Bobkov, Andrey; Hitosugi, Taro; Zhao, Jianhua; Sergienko, Eduard

Structural basis for substrate binding, catalysis, and inhibition of cancer target mitochondrial creatine kinase by a covalent inhibitor.

共价抑制剂对癌症靶标线粒体肌酸激酶的底物结合、催化和抑制的结构基础

Demir Merve, Koepping Laura, Li Ya, Fujimoto Lynn, Bobkov Andrey, Zhao Jianhua, Hitosugi Taro, Sergienko Eduard

Inhibition of therapy-resistant and metastatic melanoma by targeting the translation initiation complex

通过靶向翻译起始复合物抑制耐药性和转移性黑色素瘤

Feng, Yongmei; Diaz-Olea, Ximena; Radaeva, Mariia; Amiri, Mehdi; Joo, Hyunjeong; Kim, Hyungsoo; Ke, Xiurong; Deshpande, Aniruddha J; Olson, Steven; Jovanovic, Predrag; Pass, Ian; Deng, Qiyun; Lazar, Ikrame; Murad, Rabi; Molinolo, Alfredo; Sergienko, Eduard; Villanueva, Jessie; Topisirovic, Ivan; Jackson, Michael; Ferrone, Cristina; Sonenberg, Nahum; Cherkasov, Artem; Ronai, Ze'ev A

LARP6 regulates the mRNA translation of fibrogenic genes in liver fibrosis

LARP6 调控肝纤维化中促纤维化基因的 mRNA 翻译

Kim, Hyun Young; Mizrahi, Orel; Lee, Wonseok; Rosenthal, Sara B; Han, Cuijuan; Yee, Brian A; Blue, Steven M; Diaz, Jesiel; Jonnalagadda, Jyotiprakash; Hokutan, Kanani; Jang, Haeum; Ma, Chen-Ting; Bobkov, Andrey; Sergienko, Eduard; Jackson, Michael R; Stefanovic, Branko; Kisseleva, Tatiana; Yeo, Gene W; Brenner, David A

CD33 and clusterin interact biophysically and genetically to modulate Alzheimer risk

CD33 和簇蛋白在生物物理和遗传学上相互作用,从而调节阿尔茨海默病风险。

Dodd, Roger B; Enomoto, Masahiro; Zhou, Ye; Satoh, Kanayo; Zhang, Yalun; Chen, Fusheng; Acheson, Beatrice; Ghaffari, Deniz; Sayn-Wittgenstein, Elizabeth; Manning, Jamie J; Dukas, George V; Patel, Ronak; Burguete, Alondra Schweizer; Kralovec, Mason J; Rashid, Mamunur; Hall, Jennifer L; Tamucci, Kirstin A; Chatila, Zena K; Liu, Minghua; Lee, Annie J; Vardarajan, Badri N; Taga, Mariko F; Pollari, Sirkku; Rabinovitch, Alon; Rillahan, Cory D; Bobkov, Andrey A; Sergienko, Eduard; Meadows, William; Qamar, Seema; Randle, Suzanne J; Johnson, Christopher M; Sevalle, Jean; Griffin, Jennifer; Bohm, Christopher; Ikura, Mitsuhiko; Xian, Xunde; Herz, Joachim; Kelly, Megan A; West, Jennifer; Satapathy, Sandeep; Wilson, Mark R; Javitch, Jonathan A; Fraser, Paul E; Bennett, David A; De Jager, Philip L; Fishelson, Zvi; Frenkel, Dan; Asher, Wesley B; Bradshaw, Elizabeth M; St George-Hyslop, Peter

Novel Antimycobacterial Compounds Suppress NAD Biogenesis by Targeting a Unique Pocket of NaMN Adenylyltransferase

新型抗分枝杆菌化合物通过靶向NaMN腺苷酰转移酶的独特口袋抑制NAD生物合成

Osterman, Andrei L; Rodionova, Irina; Li, Xiaoqing; Sergienko, Eduard; Ma, Chen-Ting; Catanzaro, Antonino; Pettigrove, Mark E; Reed, Robert W; Gupta, Rashmi; Rohde, Kyle H; Korotkov, Konstantin V; Sorci, Leonardo

Discovery of 5-((5-chloro-2-methoxyphenyl)sulfonamido)nicotinamide (SBI-425), a potent and orally bioavailable tissue-nonspecific alkaline phosphatase (TNAP) inhibitor

发现 5-((5-氯-2-甲氧基苯基)磺酰胺基)烟酰胺 (SBI-425),一种强效且口服生物利用度高的组织非特异性碱性磷酸酶 (TNAP) 抑制剂

Pinkerton, Anthony B; Sergienko, Eduard; Bravo, Yalda; Dahl, Russell; Ma, Chen-Ting; Sun, Qing; Jackson, Michael R; Cosford, Nicholas D P; Millán, José Luis

TGR5 contributes to hepatic cystogenesis in rodents with polycystic liver diseases through cyclic adenosine monophosphate/Gαs signaling

TGR5通过环磷酸腺苷/Gαs信号通路促进多囊肝病啮齿动物的肝囊肿形成。

Masyuk, Tatyana V; Masyuk, Anatoliy I; Lorenzo Pisarello, Maria; Howard, Brynn N; Huang, Bing Q; Lee, Pui-Yuen; Fung, Xavier; Sergienko, Eduard; Ardecky, Robert J; Chung, Thomas D Y; Pinkerton, Anthony B; LaRusso, Nicholas F

Ectopic calcification in pseudoxanthoma elasticum responds to inhibition of tissue-nonspecific alkaline phosphatase

假性黄色瘤中的异位钙化对组织非特异性碱性磷酸酶抑制剂有反应

Ziegler, Shira G; Ferreira, Carlos R; MacFarlane, Elena Gallo; Riddle, Ryan C; Tomlinson, Ryan E; Chew, Emily Y; Martin, Ludovic; Ma, Chen-Ting; Sergienko, Eduard; Pinkerton, Anthony B; Millán, José Luis; Gahl, William A; Dietz, Harry C