日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Critical assessment of LC3/GABARAP ligands used for degrader development and ligandability of LC3/GABARAP binding pockets

对用于降解剂开发的 LC3/GABARAP 配体和 LC3/GABARAP 结合位点的配体能力进行严格评估

Martin P Schwalm, Johannes Dopfer, Adarsh Kumar, Francesco A Greco, Nicolas Bauer, Frank Löhr, Jan Heering, Sara Cano-Franco, Severin Lechner, Thomas Hanke, Ivana Jaser, Viktoria Morasch, Christopher Lenz, Daren Fearon, Peter G Marples, Charles W E Tomlinson, Lorene Brunello, Krishna Saxena, Nathan

Decrypting lysine deacetylase inhibitor action and protein modifications by dose-resolved proteomics

通过剂量分辨蛋白质组学解密赖氨酸脱乙酰酶抑制剂作用和蛋白质修饰

Yun-Chien Chang, Christian Gnann, Raphael R Steimbach, Florian P Bayer, Severin Lechner, Amirhossein Sakhteman, Miriam Abele, Jana Zecha, Jakob Trendel, Matthew The, Emma Lundberg, Aubry K Miller, Bernhard Kuster

Chemoproteomic target deconvolution reveals Histone Deacetylases as targets of (R)-lipoic acid

化学蛋白质组学靶标反卷积揭示组蛋白去乙酰化酶是 (R)-硫辛酸的靶标

Severin Lechner, Raphael R Steimbach, Longlong Wang, Marshall L Deline, Yun-Chien Chang, Tobias Fromme, Martin Klingenspor, Patrick Matthias, Aubry K Miller, Guillaume Médard, Bernhard Kuster

High-Throughput Screening and Proteomic Characterization of Compounds Targeting Myeloid-Derived Suppressor Cells

靶向髓系来源抑制细胞的化合物的高通量筛选和蛋白质组学表征

Johannes Krumm ,Elissaveta Petrova ,Severin Lechner ,Julia Mergner ,Hans-Henning Boehm ,Alessandro Prestipino ,Dominik Steinbrunn ,Marshall L Deline ,Lisa Koetzner ,Christina Schindler ,Laura Helming ,Tobias Fromme ,Martin Klingenspor ,Hannes Hahne ,Jan-Carsten Pieck ,Bernhard Kuster

Target deconvolution of HDAC pharmacopoeia reveals MBLAC2 as common off-target

HDAC 药典的靶标反卷积显示 MBLAC2 是常见的脱靶

Severin Lechner, Martin Ian P Malgapo, Christian Grätz, Raphael R Steimbach, Agnes Baron, Patrick Rüther, Simon Nadal, Carmen Stumpf, Christina Loos, Xin Ku, Polina Prokofeva, Ludwig Lautenbacher, Tino Heimburg, Vivian Würf, Chen Meng, Mathias Wilhelm, Wolfgang Sippl, Karin Kleigrewe, Josch K Paulin