日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

EXO1 promotes the meiotic MLH1-MLH3 endonuclease through conserved interactions with MLH1, MSH4 and DNA.

EXO1 通过与 MLH1、MSH4 和 DNA 的保守相互作用促进减数分裂 MLH1-MLH3 核酸内切酶

Roy Megha, Sanchez Aurore, Guerois Raphael, Senoussi Issam, Cerana Arianna, Sgrignani Jacopo, Cavalli Andrea, Rinaldi Andrea, Cejka Petr

AI-assisted design of ligands for lipocalin-2

人工智能辅助设计脂质运载蛋白-2的配体

Sgrignani, Jacopo; Buscarini, Sara; Locatelli, Patrizia; Guerra, Concetta; Furlan, Alberto; Chen, Yingyi; Zoppi, Giada; Cavalli, Andrea

FYCO1 Peptide Analogs: Design and Characterization of Autophagy Inhibitors as Co-Adjuvants in Taxane Chemotherapy of Prostate Cancer.

FYCO1肽类似物:自噬抑制剂的设计和表征,作为前列腺癌紫杉烷化疗的辅助药物

Fassi Enrico Mario Alessandro, Moretti Roberta Manuela, Montagnani Marelli Marina, Garofalo Mariangela, Gori Alessandro, Pesce Cristiano, Albani Marco, Milano Erica Ginevra, Sgrignani Jacopo, Cavalli Andrea, Grazioso Giovanni

A potent nonapeptide inhibitor for the CXCL12/HMGB1 heterocomplex: A computational and experimental approach

一种强效的 CXCL12/HMGB1 异源复合物九肽抑制剂:计算和实验方法

Fassi, Enrico Mario Alessandro; Pirani, Edisa; Cecchinato, Valentina; Cavalli, Andrea; Roda, Gabriella; Uguccioni, Mariagrazia; Sgrignani, Jacopo; Grazioso, Giovanni

A first-in-class Wiskott-Aldrich syndrome protein activator with antitumor activity in hematologic cancers

一种首创的Wiskott-Aldrich综合征蛋白激活剂,对血液肿瘤具有抗肿瘤活性

Spriano, Filippo; Sartori, Giulio; Sgrignani, Jacopo; Barnabei, Laura; Arribas, Alberto J; Guala, Matilde; Del Amor, Ana Maria Carrasco; Tomasso, Meagan R; Tarantelli, Chiara; Cascione, Luciano; Golino, Gaetanina; Riveiro, Maria E; Bortolozzi, Roberta; Lupia, Antonio; Paduano, Francesco; Huguet, Samuel; Rezai, Keyvan; Rinaldi, Andrea; Margheriti, Francesco; Ventura, Pedro; Guarda, Greta; Costa, Giosuè; Rocca, Roberta; Furlan, Alberto; Verdonk, Luuk M; Innocenti, Paolo; Martin, Nathaniel I; Viola, Giampietro; Driessen, Christoph; Zucca, Emanuele; Stathis, Anastasios; Gahtory, Digvijay; Van den Nieuwboer, Maurits; Bornhauser, Beat; Alcaro, Stefano; Trapasso, Francesco; Cristobal, Susana; Padrick, Shae B; Pazzi, Natalina; Cavalli, Franco; Cavalli, Andrea; Gaudio, Eugenio; Bertoni, Francesco

PI3Kδ activation, IL-6 overexpression, and CD37 loss cause resistance to naratuximab emtansine in lymphomas

PI3Kδ激活、IL-6过表达和CD37缺失导致淋巴瘤对那拉妥昔单抗-美坦新产生耐药性

Arribas, Alberto J; Napoli, Sara; Gaudio, Eugenio; Herbaux, Charles; Cannas, Eleonora; Tarantelli, Chiara; Bordone-Pittau, Roberta; Cascione, Luciano; Munz, Nicolas; Aresu, Luca; Sgrignani, Jacopo; Rinaldi, Andrea; Kwee, Ivo; Rossi, Davide; Cavalli, Andrea; Zucca, Emanuele; Stussi, Georg; Stathis, Anastasios; Sloss, Callum; Davids, Matthew S; Bertoni, Francesco

Esmethadone-HCl (REL-1017): a promising rapid antidepressant

盐酸艾司美沙酮(REL-1017):一种有前景的速效抗抑郁药

Fava, Maurizio; Stahl, Stephen M; De Martin, Sara; Mattarei, Andrea; Bettini, Ezio; Comai, Stefano; Alimonti, Andrea; Bifari, Francesco; Pani, Luca; Folli, Franco; Guidetti, Clotilde; Furlan, Alberto; Sgrignani, Jacopo; Locatelli, Patrizia; Cavalli, Andrea; O'Gorman, Cedric; Traversa, Sergio; Inturrisi, Charles E; Pappagallo, Marco; Manfredi, Paolo L

Machine learning analyses of antibody somatic mutations predict immunoglobulin light chain toxicity

利用机器学习分析抗体体细胞突变可以预测免疫球蛋白轻链毒性

Garofalo, Maura; Piccoli, Luca; Romeo, Margherita; Barzago, Maria Monica; Ravasio, Sara; Foglierini, Mathilde; Matkovic, Milos; Sgrignani, Jacopo; De Gasparo, Raoul; Prunotto, Marco; Varani, Luca; Diomede, Luisa; Michielin, Olivier; Lanzavecchia, Antonio; Cavalli, Andrea

How Computational Chemistry and Drug Delivery Techniques Can Support the Development of New Anticancer Drugs

计算化学和药物递送技术如何助力新型抗癌药物的研发

Garofalo, Mariangela; Grazioso, Giovanni; Cavalli, Andrea; Sgrignani, Jacopo

Isonitrile-Based Multicomponent Synthesis of β-Amino Boronic Acids as β-Lactamase Inhibitors

异腈基多组分合成β-氨基硼酸作为β-内酰胺酶抑制剂

Bassini, Emanuele; Gazzotti, Stefano; Sannio, Filomena; Presti, Leonardo Lo; Sgrignani, Jacopo; Docquier, Jean-Denis; Grazioso, Giovanni; Silvani, Alessandra