日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The multi-CDK inhibitor dinaciclib reverses bromo- and extra-terminal domain (BET) inhibitor resistance in acute myeloid leukemia via inhibition of Wnt/β-catenin signaling

多 CDK 抑制剂 dinaciclib 通过抑制 Wnt/β-catenin 信号传导逆转急性髓系白血病中溴和额外末端结构域 (BET) 抑制剂的耐药性

Alexander R Marr, Madeline Halpin, Dominique L Corbin, Yerdanos Asemelash, Steven Sher, Britten K Gordon, Ethan C Whipp, Shaneice Mitchell, Bonnie K Harrington, Shelley Orwick, Samon Benrashid, Virginia M Goettl, Vedat Yildiz, Andrew D Mitchell, Olivia Cahn, Alice S Mims, Karilyn T M Larkin, Meixao

Targeting DNA Damage Repair Functions of Two Histone Deacetylases, HDAC8 and SIRT6, Sensitizes Acute Myeloid Leukemia to NAMPT Inhibition

靶向两种组蛋白去乙酰化酶 HDAC8 和 SIRT6 的 DNA 损伤修复功能,增强急性髓系白血病对 NAMPT 抑制的敏感性

Pu Zhang, Lindsey T Brinton, Katie Williams, Steven Sher, Shelley Orwick, Lai Tzung-Huei, Alice S Mims, Christopher C Coss, Samuel K Kulp, Youssef Youssef, Wing Keung Chan, Shaneice Mitchell, Allison Mustonen, Matthew Cannon, Hannah Phillips, Amy M Lehman, Tierney Kauffman, Larry Beaver, Daniel Canf

Preclinical efficacy for a novel tyrosine kinase inhibitor, ArQule 531 against acute myeloid leukemia

新型酪氨酸激酶抑制剂 ArQule 531 治疗急性髓系白血病的临床前疗效

Ola A Elgamal, Abeera Mehmood, Jae Yoon Jeon, Bridget Carmichael, Amy Lehman, Shelley J Orwick, Jean Truxall, Virginia M Goettl, Ronni Wasmuth, Minh Tran, Shaneice Mitchell, Rosa Lapalombella, Sudharshan Eathiraj, Brian Schwartz, Kimberly Stegmaier, Sharyn D Baker, Erin Hertlein, John C Byrd

BRD4 Profiling Identifies Critical Chronic Lymphocytic Leukemia Oncogenic Circuits and Reveals Sensitivity to PLX51107, a Novel Structurally Distinct BET Inhibitor

BRD4 分析可识别关键的慢性淋巴细胞白血病致癌回路并揭示对 PLX51107(一种新型结构独特的 BET 抑制剂)的敏感性

Hatice Gulcin Ozer #, Dalia El-Gamal #, Ben Powell #, Zachary A Hing, James S Blachly, Bonnie Harrington, Shaneice Mitchell, Nicole R Grieselhuber, Katie Williams, Tzung-Huei Lai, Lapo Alinari, Robert A Baiocchi, Lindsey Brinton, Elizabeth Baskin, Matthew Cannon, Larry Beaver, Virginia M Goettl, Dav