日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Preclinical characterization of a non-peptidomimetic HIV protease inhibitor with improved metabolic stability

具有改善代谢稳定性的非肽模拟 HIV 蛋白酶抑制剂的临床前表征

Andrew Mulato, Eric Lansdon, Ron Aoyama, Johannes Voigt, Michael Lee, Albert Liclican, Gary Lee, Eric Singer, Brian Stafford, Ruoyu Gong, Bernard Murray, Julie Chan, Johnny Lee, Yili Xu, Shekeba Ahmadyar, Ana Gonzalez, Aesop Cho, George J Stepan, Uli Schmitz, Brian Schultz, Bruno Marchand, Boris Bru

A highly potent long-acting small-molecule HIV-1 capsid inhibitor with efficacy in a humanized mouse model

一种高效长效小分子 HIV-1 衣壳抑制剂,在人源化小鼠模型中有效

Stephen R Yant, Andrew Mulato, Derek Hansen, Winston C Tse, Anita Niedziela-Majka, Jennifer R Zhang, George J Stepan, Debi Jin, Melanie H Wong, Jill M Perreira, Eric Singer, Giuseppe A Papalia, Eric Y Hu, Jim Zheng, Bing Lu, Scott D Schroeder, Kevin Chou, Shekeba Ahmadyar, Albert Liclican, Helen Yu,

Abyssomicin 2 reactivates latent HIV-1 by a PKC- and HDAC-independent mechanism

Abyssomicin 2 通过一种不依赖于 PKC 和 HDAC 的机制重新激活潜伏的 HIV-1。

León, Brian; Navarro, Gabriel; Dickey, Bailey J; Stepan, George; Tsai, Angela; Jones, Gregg S; Morales, Monica E; Barnes, Tiffany; Ahmadyar, Shekeba; Tsiang, Manuel; Geleziunas, Romas; Cihlar, Tomas; Pagratis, Nikos; Tian, Yang; Yu, Helen; Linington, Roger G

Role of Mitochondrial RNA Polymerase in the Toxicity of Nucleotide Inhibitors of Hepatitis C Virus

线粒体 RNA 聚合酶在丙型肝炎病毒核苷酸抑制剂毒性中的作用

Joy Y Feng, Yili Xu, Ona Barauskas, Jason K Perry, Shekeba Ahmadyar, George Stepan, Helen Yu, Darius Babusis, Yeojin Park, Krista McCutcheon, Michel Perron, Brian E Schultz, Roman Sakowicz, Adrian S Ray