Catalytic inhibition of KAT6/KAT7 enhances the efficacy and overcomes primary and acquired resistance to Menin inhibitors in MLL leukaemia
KAT6/KAT7 的催化抑制可增强 MLL 白血病中 Menin 抑制剂的疗效并克服其原发性和获得性耐药性。
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doi:10.1101/2024.12.11.627663
Gordon, Shellaina J V; Perner, Florian; MacPherson, Laura; Wenge, Daniela V; Bourgeois, Wallace; Fennell, Katie; Klaus, Tabea; Petrovic, Jelena; Horvath, Jakub; Cao, Joan; Lapek, John; Uryu, Sean; White, Jeffrey; Lam, Enid Y N; Mu, Xinmeng Jasmine; Chan, Yih-Chih; Gillespie, Andrea; Blyth, Benjamin; Camerino, Michelle A; Bozikis, Ylyva E; Holze, Henrietta; Knezevic, Kathy; Balic, Jesse; Stupple, Paul A; Street, Ian P; Monahan, Brendon J; Sharma, Shikhar; Wainwright, Elanor N; Vassiliadis, Dane; Paul, Thomas A; Armstrong, Scott A; Dawson, Mark A