日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Association of Combination of Conformation-Specific KIT Inhibitors With Clinical Benefit in Patients With Refractory Gastrointestinal Stromal Tumors: A Phase 1b/2a Nonrandomized Clinical Trial

构象特异性KIT抑制剂联合治疗难治性胃肠道间质瘤患者的临床获益:一项1b/2a期非随机临床试验

Wagner, Andrew J; Severson, Paul L; Shields, Anthony F; Patnaik, Amita; Chugh, Rashmi; Tinoco, Gabriel; Wu, Guoxian; Nespi, Marika; Lin, Jack; Zhang, Ying; Ewing, Todd; Habets, Gaston; Burton, Elizabeth A; Matusow, Bernice; Tsai, James; Tsang, Garson; Shellooe, Rafe; Carias, Heidi; Chan, Katrina; Rezaei, Hamid; Sanftner, Laura; Marimuthu, Adhirai; Spevak, Wayne; Ibrahim, Prabha N; Inokuchi, Kerry; Alcantar, Oscar; Michelson, Glenn; Tsiatis, Athanasios C; Zhang, Chao; Bollag, Gideon; Trent, Jonathan C; Tap, William D

The RUNX1/IL-34/CSF-1R axis is an autocrinally regulated modulator of resistance to BRAF-V600E inhibition in melanoma

RUNX1/IL-34/CSF-1R 轴是黑色素瘤中对 BRAF-V600E 抑制产生抗性的自分泌调节因子

Orsi Giricz, Yongkai Mo, Kimberly B Dahlman, Xiomaris M Cotto-Rios, Chiara Vardabasso, Hoa Nguyen, Bernice Matusow, Matthias Bartenstein, Veronika Polishchuk, Douglas B Johnson, Tushar D Bhagat, Rafe Shellooe, Elizabeth Burton, James Tsai, Chao Zhang, Gaston Habets, John M Greally, Yiting Yu, Paraic

RAF inhibitors that evade paradoxical MAPK pathway activation

逃避矛盾的 MAPK 通路激活的 RAF 抑制剂

Chao Zhang, Wayne Spevak, Ying Zhang, Elizabeth A Burton, Yan Ma, Gaston Habets, Jiazhong Zhang, Jack Lin, Todd Ewing, Bernice Matusow, Garson Tsang, Adhirai Marimuthu, Hanna Cho, Guoxian Wu, Weiru Wang, Daniel Fong, Hoa Nguyen, Songyuan Shi, Patrick Womack, Marika Nespi, Rafe Shellooe, Heidi Carias

Characterizing and Overriding the Structural Mechanism of the Quizartinib-Resistant FLT3 "Gatekeeper" F691L Mutation with PLX3397

使用 PLX3397 表征和克服 Quizartinib 耐药 FLT3“守门人”F691L 突变的结构机制

Catherine C Smith, Chao Zhang, Kimberly C Lin, Elisabeth A Lasater, Ying Zhang, Evan Massi, Lauren E Damon, Matthew Pendleton, Ali Bashir, Robert Sebra, Alexander Perl, Andrew Kasarskis, Rafe Shellooe, Garson Tsang, Heidi Carias, Ben Powell, Elizabeth A Burton, Bernice Matusow, Jiazhong Zhang, Wayne

Design and pharmacology of a highly specific dual FMS and KIT kinase inhibitor

高特异性双重FMS和KIT激酶抑制剂的设计和药理学研究

Zhang, Chao; Ibrahim, Prabha N; Zhang, Jiazhong; Burton, Elizabeth A; Habets, Gaston; Zhang, Ying; Powell, Ben; West, Brian L; Matusow, Bernice; Tsang, Garson; Shellooe, Rafe; Carias, Heidi; Nguyen, Hoa; Marimuthu, Adhirai; Zhang, Kam Y J; Oh, Angela; Bremer, Ryan; Hurt, Clarence R; Artis, Dean R; Wu, Guoxian; Nespi, Marika; Spevak, Wayne; Lin, Paul; Nolop, Keith; Hirth, Peter; Tesch, Greg H; Bollag, Gideon

A strategy for constructing aneuploid yeast strains by transient nondisjunction of a target chromosome

利用靶染色体的瞬时不分离构建非整倍体酵母菌株的策略

Anders, Kirk R; Kudrna, Julie R; Keller, Kirstie E; Kinghorn, BreAnna; Miller, Elizabeth M; Pauw, Daniel; Peck, Anders T; Shellooe, Christopher E; Strong, Isaac J T