Pre-clinical pharmacology and mechanism of action of SG3199, the pyrrolobenzodiazepine (PBD) dimer warhead component of antibody-drug conjugate (ADC) payload tesirine
SG3199(抗体-药物偶联物 (ADC) 有效载荷 tesirine 的吡咯并苯二氮卓 (PBD) 二聚体弹头组分)的临床前药理学和作用机制
期刊:Scientific Reports
影响因子:3.8
doi:10.1038/s41598-018-28533-4
John A Hartley, Michael J Flynn, John P Bingham, Simon Corbett, Halla Reinert, Arnaud Tiberghien, Luke A Masterson, Dyeison Antonow, Lauren Adams, Sajidah Chowdhury, David G Williams, Shenlan Mao, Jay Harper, Carin E G Havenith, Francesca Zammarchi, Simon Chivers, Patrick H van Berkel, Philip W Howa