日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural Modifications Reveal Dual Functions of the C-4 Carbonyl Group in the Fatty Acid Chain of Ipomoeassin F

结构修饰揭示了番薯素F脂肪酸链中C-4羰基的双重功能

Khosravi, Arman; Nnamdi, Precious; May, Alexa; Slattery, Kelsey; Sammelson, Robert E; Shi, Wei Q

Effect of Ipomoeassin F on the Synthesis of Membrane and Secretory Proteins in Triple-Negative Breast Cancer Cells.

番薯素F对三阴性乳腺癌细胞膜蛋白和分泌蛋白合成的影响

Sicairos Brihget, Zhou Jianhong, Hu Zhijian, Zhang Qingyang, Shi Wei Q, Du Yuchun

Synthesis, Biological Evaluation and Docking Studies of Ring-Opened Analogues of Ipomoeassin F

番薯素F开环类似物的合成、生物学评价和分子对接研究

O'Keefe, Sarah; Bhadra, Pratiti; Duah, Kwabena B; Zong, Guanghui; Tenay, Levise; Andrews, Lauren; Schneider, Hayden; Anderson, Ashley; Hu, Zhijian; Aljewari, Hazim S; Hall, Belinda S; Simmonds, Rachel E; Helms, Volkhard; High, Stephen; Shi, Wei Q

Ipomoeassin F Binds Sec61α to Inhibit Protein Translocation

番薯素F与Sec61α结合以抑制蛋白质转位

Zong, Guanghui; Hu, Zhijian; O'Keefe, Sarah; Tranter, Dale; Iannotti, Michael J; Baron, Ludivine; Hall, Belinda; Corfield, Katherine; Paatero, Anja O; Henderson, Mark J; Roboti, Peristera; Zhou, Jianhong; Sun, Xianwei; Govindarajan, Mugunthan; Rohde, Jason M; Blanchard, Nicolas; Simmonds, Rachel; Inglese, James; Du, Yuchun; Demangel, Caroline; High, Stephen; Paavilainen, Ville O; Shi, Wei Q

Simultaneous Targeting of NPC1 and VDAC1 by Itraconazole Leads to Synergistic Inhibition of mTOR Signaling and Angiogenesis

伊曲康唑同时靶向NPC1和VDAC1可协同抑制mTOR信号通路和血管生成

Head, Sarah A; Shi, Wei Q; Yang, Eun Ju; Nacev, Benjamin A; Hong, Sam Y; Pasunooti, Kalyan K; Li, Ruo-Jing; Shim, Joong Sup; Liu, Jun O

Design, synthesis and biological evaluation of fucose-truncated monosaccharide analogues of ipomoeassin F

番薯素F的岩藻糖截短单糖类似物的设计、合成和生物学评价

Zong, Guanghui; Hirsch, Melissa; Mondrik, Collin; Hu, Zhijian; Shi, Wei Q

Revealing the Pharmacophore of Ipomoeassin F through Molecular Editing

通过分子编辑揭示番薯素F的药效团

Zong, Guanghui; Aljewari, Hazim; Hu, Zhijian; Shi, Wei Q