日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery and dynamic pharmacology of μ-opioid receptor positive allosteric modulators

μ-阿片受体正向变构调节剂的发现和动态药理学

O'Brien, Evan S; Wang, Junzheng; Tanguturi, Parthasaradhireddy; Li, Mengchu; White, Elizabeth; Shiimura, Yuki; Paul, Barnali; Appourchaux, Kevin; Kumar, Kaavya Krishna; Huang, Weijiao; Majumdar, Susruta; Traynor, John R; Streicher, John M; Chen, Chunlai; Kobilka, Brian K

A cryptic pocket in CB1 drives peripheral and functional selectivity

CB1 中的一个隐蔽口袋驱动外周和功能选择性

Rangari, Vipin Ashok; O'Brien, Evan S; Powers, Alexander S; Slivicki, Richard A; Bertels, Zachariah; Appourchaux, Kevin; Aydin, Deniz; Ramos-Gonzalez, Nokomis; Mwirigi, Juliet; Lin, Li; Mangutov, Elizaveta; Sobecks, Briana L; Awad-Agbaria, Yaseen; Uphade, Manoj B; Aguilar, Jhoan; Peddada, Teja Nikhil; Shiimura, Yuki; Huang, Xi-Ping; Folarin-Hines, Jakayla; Payne, Maria; Kalathil, Anirudh; Varga, Balazs R; Kobilka, Brian K; Pradhan, Amynah A; Cameron, Michael D; Kumar, Kaavya Krishna; Dror, Ron O; Gereau, Robert W 4th; Majumdar, Susruta

Virtual library docking for cannabinoid-1 receptor agonists with reduced side effects.

针对副作用较小的 1 型大麻素受体激动剂的虚拟库对接

Tummino Tia A, Iliopoulos-Tsoutsouvas Christos, Braz Joao M, O'Brien Evan S, Stein Reed M, Craik Veronica, Tran Ngan K, Ganapathy Suthakar, Liu Fangyu, Shiimura Yuki, Tong Fei, Ho Thanh C, Radchenko Dmytro S, Moroz Yurii S, Rosado Sian Rodriguez, Bhardwaj Karnika, Benitez Jorge, Liu Yongfeng, Kandasamy Herthana, Normand Claire, Semache Meriem, Sabbagh Laurent, Glenn Isabella, Irwin John J, Kumar Kaavya Krishna, Makriyannis Alexandros, Basbaum Allan I, Shoichet Brian K

How the ghrelin receptor recognizes the acyl-modified orexigenic hormone

胃饥饿素受体如何识别酰基修饰的促食欲激素

Shiimura, Yuki; Kojima, Masayasu; Sato, Takahiro

Ghrelin-LEAP2 interactions along the stomach-liver axis

胃-肝轴上的生长素释放肽-LEAP2相互作用

Sakai, Katsuya; Nakazato, Yuki; Shiimura, Yuki; Zhang, Weidong; Nakazato, Masamitsu

A µ-opioid receptor modulator that works cooperatively with naloxone.

一种与纳洛酮协同作用的μ-阿片受体调节剂

O'Brien Evan S, Rangari Vipin Ashok, El Daibani Amal, Eans Shainnel O, Hammond Haylee R, White Elizabeth, Wang Haoqing, Shiimura Yuki, Krishna Kumar Kaavya, Jiang Qianru, Appourchaux Kevin, Huang Weijiao, Zhang Chensong, Kennedy Brandon J, Mathiesen Jesper M, Che Tao, McLaughlin Jay P, Majumdar Susruta, Kobilka Brian K

Acyl modifications in bovine, porcine, and equine ghrelins

牛、猪和马生长素释放肽的酰基修饰

Ida, Takanori; Tominaga, Hatsumi; Iwamoto, Eri; Kurogi, Akito; Okura, Ayaka; Shimada, Kengo; Kato, Johji; Kuwano, Atsutoshi; Ode, Hirotaka; Nagata, Sayaka; Kitamura, Kazuo; Yazawa, Takashi; Sato-Hashimoto, Miho; Yasuda, Masahiro; Miyazato, Mikiya; Shiimura, Yuki; Sato, Takahiro; Kojima, Masayasu

Large library docking for cannabinoid-1 receptor agonists with reduced side effects

针对副作用较小的1型大麻素受体激动剂的大型化合物库对接

Tummino, Tia A; Iliopoulos-Tsoutsouvas, Christos; Braz, Joao M; O'Brien, Evan S; Stein, Reed M; Craik, Veronica; Tran, Ngan K; Ganapathy, Suthakar; Liu, Fangyu; Shiimura, Yuki; Tong, Fei; Ho, Thanh C; Radchenko, Dmytro S; Moroz, Yurii S; Rosado, Sian Rodriguez; Bhardwaj, Karnika; Benitez, Jorge; Liu, Yongfeng; Kandasamy, Herthana; Normand, Claire; Semache, Meriem; Sabbagh, Laurent; Glenn, Isabella; Irwin, John J; Kumar, Kaavya Krishna; Makriyannis, Alexandros; Basbaum, Allan I; Shoichet, Brian K

Structural insights into the agonists binding and receptor selectivity of human histamine H(4) receptor

人组胺H(4)受体激动剂结合及受体选择性的结构解析

Im, Dohyun; Kishikawa, Jun-Ichi; Shiimura, Yuki; Hisano, Hiromi; Ito, Akane; Fujita-Fujiharu, Yoko; Sugita, Yukihiko; Noda, Takeshi; Kato, Takayuki; Asada, Hidetsugu; Iwata, So

Insights Into the Regulation of Offspring Growth by Maternally Derived Ghrelin

母源性生长素释放肽对后代生长调控的深入研究

Sato, Takahiro; Ida, Takanori; Shiimura, Yuki; Matsui, Kazuma; Oishi, Kanae; Kojima, Masayasu