日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery and Characterization of the Potent and Highly Selective 1,7-Naphthyridine-Based Inhibitors BAY-091 and BAY-297 of the Kinase PIP4K2A

发现并表征强效且高选择性的 1,7-萘啶类激酶 PIP4K2A 抑制剂 BAY-091 和 BAY-297

Lars Wortmann, Nico Bräuer, Simon J Holton, Horst Irlbacher, Jörg Weiske, Christian Lechner, Robin Meier, Jakob Karén, Catrine Berthold Siöberg, Vera Pütter, Clara D Christ, Antonius Ter Laak, Philip Lienau, Ralf Lesche, Barbara Nicke, Shing-Hu Cheung, Marcus Bauser, Andrea Haegebarth, Franz von Nus

RAF dimer inhibition enhances the antitumor activity of MEK inhibitors in K-RAS mutant tumors

RAF 二聚体抑制可增强 MEK 抑制剂在 K-RAS 突变肿瘤中的抗肿瘤活性

Xi Yuan, Zhiyu Tang, Rong Du, Zhan Yao, Shing-Hu Cheung, Xinwen Zhang, Jing Wei, Yuan Zhao, Yunguang Du, Ye Liu, Xiaoxia Hu, Wenfeng Gong, Yong Liu, Yajuan Gao, Zhiyue Huang, Zongfu Cao, Min Wei, Changyou Zhou, Lai Wang, Neal Rosen, Paul D Smith, Lusong Luo

ADTRP regulates TFPI expression via transcription factor POU1F1 involved in coronary artery disease

ADTRP 通过转录因子 POU1F1 调节与冠状动脉疾病有关的 TFPI 表达

Chunyan Luo, Elisabeth Pook, Fan Wang, Stephen R Archacki, Bo Tang, Weiyi Zhang, Jing-Shan Hu, Jian Yang, Kirsten Leineweber, Martin Bechem, Weifeng Huang, Yinhong Song, Shing-Hu Cheung, Volker Laux, Tie Ke, Xiang Ren, Xin Tu, Qiuyun Chen, Qing Kenneth Wang, Chengqi Xu

Androgen inhibits key atherosclerotic processes by directly activating ADTRP transcription

雄激素通过直接激活 ADTRP 转录来抑制关键动脉粥样硬化过程

Chunyan Luo, Elisabeth Pook, Bo Tang, Weiyi Zhang, Sisi Li, Kirsten Leineweber, Shing-Hu Cheung, Qiuyun Chen, Martin Bechem, Jing-Shan Hu, Volker Laux, Qing Kenneth Wang

BGB-283, a Novel RAF Kinase and EGFR Inhibitor, Displays Potent Antitumor Activity in BRAF-Mutated Colorectal Cancers

BGB-283 是一种新型 RAF 激酶和 EGFR 抑制剂,在 BRAF 突变的结肠直肠癌中表现出强大的抗肿瘤活性

Zhiyu Tang, Xi Yuan, Rong Du, Shing-Hu Cheung, Guoliang Zhang, Jing Wei, Yuan Zhao, Yingcai Feng, Hao Peng, Yi Zhang, Yunguang Du, Xiaoxia Hu, Wenfeng Gong, Yong Liu, Yajuan Gao, Ye Liu, Rui Hao, Shengjian Li, Shaohui Wang, Jiafu Ji, Lianhai Zhang, Shuangxi Li, David Sutton, Min Wei, Changyou Zhou,