日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Small molecule-induced mitochondrial disruption directs prostate cancer inhibition via UPR signaling

小分子诱导的线粒体破坏通过 UPR 信号传导指导前列腺癌抑制

Elizabeth Rico-Bautista, Wenhong Zhu, Shinichi Kitada, Suthakar Ganapathy, Eric Lau, Stan Krajewski, Joel Ramirez, Jason A Bush, Zhimin Yuan, Dieter A Wolf

Design and characterization of a potent and selective dual ATP- and substrate-competitive subnanomolar bidentate c-Jun N-terminal kinase (JNK) inhibitor

设计和表征一种强效且选择性双重 ATP 和底物竞争性亚纳摩尔双齿 c-Jun N 端激酶 (JNK) 抑制剂

John L Stebbins, Surya K De, Petra Pavlickova, Vida Chen, Thomas Machleidt, Li-Hsing Chen, Christian Kuntzen, Shinichi Kitada, Michael Karin, Maurizio Pellecchia

Efficient elimination of cancer cells by deoxyglucose-ABT-263/737 combination therapy

脱氧葡萄糖-ABT-263/737联合疗法有效消除癌细胞

Ryuji Yamaguchi, Edith Janssen, Guy Perkins, Mark Ellisman, Shinichi Kitada, John C Reed

BI-97C1, an optically pure Apogossypol derivative as pan-active inhibitor of antiapoptotic B-cell lymphoma/leukemia-2 (Bcl-2) family proteins

BI-97C1 是一种光学纯的阿朴棉酚衍生物,可作为抗凋亡 B 细胞淋巴瘤/白血病-2 (Bcl-2) 家族蛋白的全活性抑制剂

Jun Wei, John L Stebbins, Shinichi Kitada, Rupesh Dash, William Placzek, Michele F Rega, Bainan Wu, Jason Cellitti, Dayong Zhai, Li Yang, Russell Dahl, Paul B Fisher, John C Reed, Maurizio Pellecchia

Bcl-B expression in human epithelial and nonepithelial malignancies

人类上皮和非上皮恶性肿瘤中的 Bcl-B 表达

Maryla Krajewska, Shinichi Kitada, Jane N Winter, Daina Variakojis, Alan Lichtenstein, Dayong Zhai, Michael Cuddy, Xianshu Huang, Frederic Luciano, Cheryl H Baker, Hoguen Kim, Eunah Shin, Susan Kennedy, Allen H Olson, Andrzej Badzio, Jacek Jassem, Ivo Meinhold-Heerlein, Michael J Duffy, Aaron D Schi