日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Coronary Artery Disease in Female Athletes

女性运动员的冠状动脉疾病

Kazum-Beisr, Shirit; Schamroth-Pravada, Nili; Porter, Avital; Moshe, Roi; Hamdan, Ashraf; Kornowski, Ran; Constantini, Naama

PIP4K2C inhibition reverses autophagic flux impairment induced by SARS-CoV-2.

PIP4K2C 抑制可逆转 SARS-CoV-2 引起的自噬通量受损

Karim Marwah, Mishra Manjari, Lo Chieh-Wen, Saul Sirle, Cagirici Halise Busra, Gourdelier Manon, Ghita Luca, Ojha Amrita, Tran Do Hoang Nhu, Agrawal Aditi, McGraw Connor, East Michael P, Gammeltoft Karen Anbro, Sahoo Malaya Kumar, Mooney Nancie A, Johnson Gary L, Das Soumita, Leyssen Pieter, Neyts Johan, Chiu Winston, Cohen Courtney A, Bukh Jens, Gottwein Judith, Dye John M, Neff Norma, Jackson Peter K, Pinsky Benjamin A, Laitinen Tuomo, Pantsar Tatu, Poso Antti, Zanini Fabio, De Jonghe Steven, Asquith Christopher R M, Einav Shirit

Development of pyrazolo[1,5-a]pyrimidine based macrocyclic kinase inhibitors targeting AAK1.

开发以吡唑并[1,5-a]嘧啶为基础的大环激酶抑制剂,靶向AAK1。

Mensing Theresa E, Kurz Christian G, Amrhein Jennifer A, Ehret Theresa A L, Preuss Franziska, Mathea Sebastian, Karim Marwah, Tran Do Hoang Nhu, Kadlecova Zuzana, Tolvanen Tuomas A, Martinez-Molina Daniel, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas

An orally bioavailable SARS-CoV-2 main protease inhibitor exhibits improved affinity and reduced sensitivity to mutations.

口服生物利用度高的 SARS-CoV-2 主蛋白酶抑制剂表现出更高的亲和力和更低的突变敏感性

Westberg Michael, Su Yichi, Zou Xinzhi, Huang Pinghan, Rustagi Arjun, Garhyan Jaishree, Patel Puja Bhavesh, Fernandez Daniel, Wu Yan, Hao Chenzhou, Lo Chieh-Wen, Karim Marwah, Ning Lin, Beck Aimee, Saenkham-Huntsinger Panatda, Tat Vivian, Drelich Aleksandra, Peng Bi-Hung, Einav Shirit, Tseng Chien-Te K, Blish Catherine, Lin Michael Z

Systems immunology of transcriptional responses to viral infection identifies conserved antiviral pathways across macaques and humans

系统免疫学对病毒感染转录反应的研究揭示了猕猴和人类中保守的抗病毒通路。

Ratnasiri, Kalani; Zheng, Hong; Toh, Jiaying; Yao, Zhiyuan; Duran, Veronica; Donato, Michele; Roederer, Mario; Kamath, Megha; Todd, John-Paul M; Gagne, Matthew; Foulds, Kathryn E; Francica, Joseph R; Corbett, Kizzmekia S; Douek, Daniel C; Seder, Robert A; Einav, Shirit; Blish, Catherine A; Khatri, Purvesh

Back-Pocket Optimization of 2-Aminopyrimidine-Based Macrocycles Leads to Potent EPHA2/GAK Kinase Inhibitors.

2-氨基嘧啶基大环化合物的后口袋优化可得到强效的EPHA2/GAK激酶抑制剂

Gerninghaus Joshua, Zhubi Rezart, Krämer Andreas, Karim Marwah, Tran Do Hoang Nhu, Joerger Andreas C, Schreiber Christian, Berger Lena M, Berger Benedict-Tilman, Ehret Theresa A L, Elson Lewis, Lenz Christopher, Saxena Krishna, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas

Chemical inactivation strategies for SARS-CoV-2-infected cells and organoids

SARS-CoV-2 感染细胞和类器官的化学灭活策略

Marwah Karim, Amol Arunrao Pohane, Chieh-Wen Lo, Shirit Einav, Jaishree Garhyan

Back-pocket optimization of 2-aminopyrimidine-based macrocycles leads to potent dual EPHA2/GAK kinase inhibitors with antiviral activity

对 2-氨基嘧啶大环化合物进行后袋优化,可得到具有抗病毒活性的强效双重 EPHA2/GAK 激酶抑制剂

Joshua Gerninghaus, Rezart Zhubi, Andreas Krämer, Marwah Karim, Do Hoang Nhu Tran, Andreas C Joerger, Christian Schreiber, Lena M Berger, Benedict-Tilman Berger, Theresa A L Ehret, Lewis Elson, Christopher Lenz, Krishna Saxena, Susanne Müller, Shirit Einav, Stefan Knapp, Thomas Hanke

Dynamic T-Wave Inversion: Unraveling an Athlete's Heart Mystery

动态T波倒置:揭开运动员心脏之谜

Kazum, Shirit Sara; Hoss, Sara; Monakier, Daniel; Hamdan, Ashraf; Kornowski, Ran

Single B cell transcriptomics identifies multiple isotypes of broadly neutralizing antibodies against flaviviruses

单B细胞转录组学鉴定出多种针对黄病毒的广谱中和抗体同型

Jay Lubow ,Lisa M Levoir ,Duncan K Ralph ,Laura Belmont ,Maya Contreras ,Catiana H Cartwright-Acar ,Caroline Kikawa ,Shruthi Kannan ,Edgar Davidson ,Veronica Duran ,David E Rebellon-Sanchez ,Ana M Sanz ,Fernando Rosso ,Benjamin J Doranz ,Shirit Einav ,Frederick A Matsen Iv ,Leslie Goo