Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells
强效且选择性的 KDM5 抑制剂可阻止转录起始位点的 H3K4me3 细胞去甲基化和 MM1S 骨髓瘤细胞的增殖
期刊:Cell Chemical Biology
影响因子:6.6
doi:10.1016/j.chembiol.2017.02.006
Anthony Tumber, Andrea Nuzzi, Edward S Hookway, Stephanie B Hatch, Srikannathasan Velupillai, Catrine Johansson, Akane Kawamura, Pavel Savitsky, Clarence Yapp, Aleksandra Szykowska, Na Wu, Chas Bountra, Claire Strain-Damerell, Nicola A Burgess-Brown, Gian Filippo Ruda, Oleg Fedorov, Shonagh Munro, K