日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Long non-coding RNA-derived peptides are immunogenic and drive a potent anti-tumour response

长链非编码 RNA 衍生肽具有免疫原性,可引发强效的抗肿瘤反应

Wojciech Barczak #, Simon M Carr #, Geng Liu, Shonagh Munro, Annalisa Nicastri, Lian Ni Lee, Claire Hutchings, Nicola Ternette, Paul Klenerman, Alexander Kanapin, Anastasia Samsonova, Nicholas B La Thangue

Combination treatment of T1-44, a PRMT5 inhibitor with Vactosertib, an inhibitor of TGF-β signaling, inhibits invasion and prolongs survival in a mouse model of pancreatic tumors

PRMT5 抑制剂 T1-44 与 TGF-β 信号抑制剂 Vactosertib 联合治疗可抑制小鼠胰腺肿瘤模型的侵袭并延长其生存期

Eunji Hong, Wojciech Barczak, Sujin Park, Jin Sun Heo, Akira Ooshima, Shonagh Munro, Chang Pyo Hong, Jinah Park, Haein An, Joon Oh Park, Seok Hee Park, Nick B La Thangue, Seong-Jin Kim

PRMT5 promotes cancer cell migration and invasion through the E2F pathway

PRMT5通过E2F通路促进癌细胞迁移和侵袭

Wojciech Barczak #, Li Jin #, Simon Mark Carr, Shonagh Munro, Samuel Ward, Alexander Kanapin, Anastasia Samsonova, Nicholas B La Thangue

Arginine methylation expands the regulatory mechanisms and extends the genomic landscape under E2F control

精氨酸甲基化扩展了调控机制并扩展了 E2F 控制下的基因组格局

Alice Poppy Roworth, Simon Mark Carr, Geng Liu, Wojciech Barczak, Rebecca Louise Miller, Shonagh Munro, Alexander Kanapin, Anastasia Samsonova, Nicholas B La Thangue

Functional interplay between E2F7 and ribosomal rRNA gene transcription regulates protein synthesis

E2F7 与核糖体 rRNA 基因转录之间的功能相互作用调节蛋白质合成

Amanda S Coutts, Shonagh Munro, Nicholas B La Thangue

Tudor-domain protein PHF20L1 reads lysine methylated retinoblastoma tumour suppressor protein

Tudor 结构域蛋白 PHF20L1 读取赖氨酸甲基化的视网膜母细胞瘤肿瘤抑制蛋白

Simon M Carr, Shonagh Munro, Cari A Sagum, Oleg Fedorov, Mark T Bedford, Nicholas B La Thangue

Linker Histone H1.2 Directs Genome-wide Chromatin Association of the Retinoblastoma Tumor Suppressor Protein and Facilitates Its Function

连接组蛋白 H1.2 指导视网膜母细胞瘤肿瘤抑制蛋白的全基因组染色质结合并促进其功能

Shonagh Munro, Edward S Hookway, Melanie Floderer, Simon M Carr, Rebecca Konietzny, Benedikt M Kessler, Udo Oppermann, Nicholas B La Thangue

Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells

强效且选择性的 KDM5 抑制剂可阻止转录起始位点的 H3K4me3 细胞去甲基化和 MM1S 骨髓瘤细胞的增殖

Anthony Tumber, Andrea Nuzzi, Edward S Hookway, Stephanie B Hatch, Srikannathasan Velupillai, Catrine Johansson, Akane Kawamura, Pavel Savitsky, Clarence Yapp, Aleksandra Szykowska, Na Wu, Chas Bountra, Claire Strain-Damerell, Nicola A Burgess-Brown, Gian Filippo Ruda, Oleg Fedorov, Shonagh Munro, K

Citrullination-acetylation interplay guides E2F-1 activity during the inflammatory response

瓜氨酸化-乙酰化相互作用在炎症反应过程中引导 E2F-1 活性

Fatemeh Ghari, Anne-Marie Quirke, Shonagh Munro, Joanna Kawalkowska, Sarah Picaud, Joanna McGouran, Venkataraman Subramanian, Aaron Muth, Richard Williams, Benedikt Kessler, Paul R Thompson, Panagis Fillipakopoulos, Stefan Knapp, Patrick J Venables, Nicholas B La Thangue

Selective inhibition of BET bromodomains

选择性抑制 BET 溴结构域

Panagis Filippakopoulos, Jun Qi, Sarah Picaud, Yao Shen, William B Smith, Oleg Fedorov, Elizabeth M Morse, Tracey Keates, Tyler T Hickman, Ildiko Felletar, Martin Philpott, Shonagh Munro, Michael R McKeown, Yuchuan Wang, Amanda L Christie, Nathan West, Michael J Cameron, Brian Schwartz, Tom D Height