日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Simulations and active learning enable efficient identification of an experimentally-validated broad coronavirus inhibitor.

模拟和主动学习能够有效地识别经实验验证的广谱冠状病毒抑制剂

Elez Katarina, Hempel Tim, Shrimp Jonathan H, Moor Nicole, Raich Lluís, Rocha Cheila, Winter Robin, Le Tuan, Pöhlmann Stefan, Hoffmann Markus, Hall Matthew D, Noé Frank

Mass spectrometry-guided discovery of novel GCPII inhibitor scaffolds

质谱引导下新型GCPII抑制剂骨架的发现

Wiseman, Robyn; Thomas, Ajit G; Janiszewski, John; Hoxie, Nate; Lee, Chae Bin; Wu, Ying; Tsukamoto, Takashi; Ye, Lin; Ronzetti, Michael; Shrimp, Jonathan H; Adderley, Davina; Rai, Ganesha; Rais, Rana; Alt, Jesse; Hall, Matthew D; Hu, Xin; Kales, Stephen C; Slusher, Barbara S

Methotrexate-based PROTACs as DHFR-specific chemical probes

基于甲氨蝶呤的 PROTAC 作为 DHFR 特异性化学探针

Sandeep Rana, Patricia Dranchak, Jayme L Dahlin, Laurence Lamy, Wenqing Li, Erin Oliphant, Jonathan H Shrimp, Girish H Rajacharya, Ravi Tharakan, David O Holland, Apryl S Whitten, Kelli M Wilson, Pankaj K Singh, Scott K Durum, Dingyin Tao, Ganesha Rai, James Inglese

Notes on AEMS methods development for high throughput experimentation in drug discovery

关于用于药物发现高通量实验的AEMS方法开发的说明

Verma, Meghav; Hoxie, Nate; Janiszewski, John; Bonney, Charles; Hall, Matthew D; Michael, Sam; Covey, Tom; Shrimp, Jonathan H

SULT1A1-dependent sulfonation of alkylators is a lineage-dependent vulnerability of liver cancers

SULT1A1 依赖的烷基化磺化是肝癌谱系依赖性的易感性

Lei Shi, William Shen, Mindy I Davis, Ke Kong, Phuong Vu, Supriya K Saha, Ramzi Adil, Johannes Kreuzer, Regina Egan, Tobie D Lee, Patricia Greninger, Jonathan H Shrimp, Wei Zhao, Ting-Yu Wei, Mi Zhou, Jason Eccleston, Jonathan Sussman, Ujjawal Manocha, Vajira Weerasekara, Hiroshi Kondo, Vindhya Vija

Reference compounds for characterizing cellular injury in high-content cellular morphology assays

用于在高内涵细胞形态学测定中表征细胞损伤的参考化合物

Jayme L Dahlin #, Bruce K Hua #, Beth E Zucconi, Shawn D Nelson Jr, Shantanu Singh, Anne E Carpenter, Jonathan H Shrimp, Evelyne Lima-Fernandes, Mathias J Wawer, Lawrence P W Chung, Ayushi Agrawal, Mary O'Reilly, Dalia Barsyte-Lovejoy, Magdalena Szewczyk, Fengling Li, Parnian Lak, Matthew Cuellar, P

Mitoribosome sensitivity to HSP70 inhibition uncovers metabolic liabilities of castration-resistant prostate cancer

线粒体核糖体对 HSP70 抑制的敏感性揭示了去势抵抗性前列腺癌的代谢负担

Frank J Echtenkamp, Ryo Ishida, Genesis M Rivera-Marquez, Marisa Maisiak, Oleta T Johnson, Jonathan H Shrimp, Arnav Sinha, Stephen John Ralph, Ian Nisbet, Murali Krishna Cherukuri, Jason E Gestwicki, Leonard M Neckers

Nonspecific membrane bilayer perturbations by ivermectin underlie SARS-CoV-2 in vitro activity

伊维菌素对非特异性膜双层的扰动是 SARS-CoV-2 体外活性的基础

Richard T Eastman, Radda Rusinova, Karl F Herold, Xi-Ping Huang, Patricia Dranchak, Ty C Voss, Sandeep Rana, Jonathan H Shrimp, Alex D White, Hugh C Hemmings Jr, Bryan L Roth, James Inglese, Olaf S Andersen, Jayme L Dahlin

Suite of TMPRSS2 Assays for Screening Drug Repurposing Candidates as Potential Treatments of COVID-19

TMPRSS2 检测套件可用于筛选可作为 COVID-19 潜在治疗方法的药物再利用候选药物

Jonathan H Shrimp, John Janiszewski, Catherine Z Chen, Miao Xu, Kelli M Wilson, Stephen C Kales, Philip E Sanderson, Paul Shinn, Rick Schneider, Zina Itkin, Hui Guo, Min Shen, Carleen Klumpp-Thomas, Samuel G Michael, Wei Zheng, Anton Simeonov, Matthew D Hall

A Suite of TMPRSS2 Assays for Screening Drug Repurposing Candidates as Potential Treatments of COVID-19

一套 TMPRSS2 检测试剂盒可用于筛选可作为 COVID-19 潜在治疗方法的药物再利用候选药物

Jonathan H Shrimp, John Janiszewski, Catherine Z Chen, Miao Xu, Kelli M Wilson, Stephen C Kales, Philip E Sanderson, Paul Shinn, Zina Itkin, Hui Guo, Min Shen, Carleen Klumpp-Thomas, Samuel G Michael, Wei Zheng, Anton Simeonov, Matthew D Hall