日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Non-Classical Neuroactive Steroid Exhibiting Potent, Efficacious GABA (A) Receptor Agonism and NMDA Receptor Inhibition

一种非经典神经活性类固醇,具有强效的GABA(A)受体激动作用和NMDA受体抑制作用。

Shu, Hong-Jin; Xu, Yuanjian; Qian, Mingxing; Benz, Ann; Yuede, Carla M; Covey, Douglas F; Zorumski, Charles F; Mennerick, Steven

A Role for δ Subunit-Containing GABA(A) Receptors on Parvalbumin-Positive Neurons in Maintaining Electrocortical Signatures of Sleep States.

α亚基GABA(A)受体在小白蛋白阳性神经元上的作用在维持睡眠状态的脑电皮层特征中的作用

Lambert Peter M, Salvatore Sofia V, Lu Xinguo, Shu Hong-Jin, Benz Ann, Rensing Nicholas, Yuede Carla M, Wong Michael, Zorumski Charles F, Mennerick Steven

δ-Containing GABA(A) receptors on parvalbumin interneurons modulate neuronal excitability and network dynamics in the mouse medial prefrontal cortex

小鼠内侧前额叶皮层中,小白蛋白中间神经元上的δ亚基GABA(A)受体调节神经元兴奋性和网络动力学。

Lu, Xinguo; Shu, Hong-Jin; Lambert, Peter M; Benz, Ann; Zorumski, Charles F; Mennerick, Steven

Effects of Complete and Partial Loss of the 24S-Hydroxycholesterol-Generating Enzyme Cyp46a1 on Behavior and Hippocampal Transcription in Mouse.

24S-羟基胆固醇生成酶Cyp46a1完全和部分缺失对小鼠行为和海马转录的影响

Shu Hong-Jin, Ziolkowski Luke H, Salvatore Sofia V, Benz Ann M, Wozniak David F, Yuede Carla M, Paul Steven M, Zorumski Charles F, Mennerick Steven

Synthesis and evaluation of photoaffinity labeling reagents for identifying binding sites of sulfated neurosteroids on NMDA and GABA(A) receptors

合成和评价光亲和标记试剂,用于鉴定硫酸神经甾体在NMDA和GABA(A)受体上的结合位点

Qian, Mingxing; Xu, Yuanjian; Shu, Hong-Jin; Chen, Zi-Wei; Wang, Lei; Zorumski, Charles F; Evers, Alex S; Mennerick, Steven; Covey, Douglas F

A neuroactive steroid with a therapeutically interesting constellation of actions at GABA(A) and NMDA receptors

一种具有神经活性的类固醇,对GABA(A)和NMDA受体具有治疗上有趣的多种作用。

Ziolkowski, Luke; Mordukhovich, Isaac; Chen, Daniel M; Chisari, Mariangela; Shu, Hong-Jin; Lambert, Peter M; Qian, Mingxing; Zorumski, Charles F; Covey, Douglas F; Mennerick, Steven

Effects of CYP46A1 Inhibition on Long-Term-Depression in Hippocampal Slices ex vivo and 24S-Hydroxycholesterol Levels in Mice in vivo

CYP46A1抑制对离体海马切片长期抑制及体内小鼠24S-羟基胆固醇水平的影响

Popiolek, Michael; Izumi, Yukitoshi; Hopper, Allen T; Dai, Jing; Miller, Silke; Shu, Hong-Jin; Zorumski, Charles F; Mennerick, Steven

Positive Allosteric Modulation as a Potential Therapeutic Strategy in Anti-NMDA Receptor Encephalitis

正向变构调节作为抗NMDA受体脑炎的潜在治疗策略

Warikoo, Natasha; Brunwasser, Samuel J; Benz, Ann; Shu, Hong-Jin; Paul, Steven M; Lewis, Michael; Doherty, James; Quirk, Michael; Piccio, Laura; Zorumski, Charles F; Day, Gregory S; Mennerick, Steven

Fast phasic release properties of dopamine studied with a channel biosensor

利用通道生物传感器研究多巴胺的快速相释放特性

Kress, Geraldine J; Shu, Hong-Jin; Yu, Andrew; Taylor, Amanda; Benz, Ann; Harmon, Steve; Mennerick, Steven

Photodynamic effects of steroid-conjugated fluorophores on GABAA receptors

类固醇偶联荧光团对GABAA受体的光动力学效应

Shu, Hong-Jin; Eisenman, Lawrence N; Wang, Cunde; Bandyopadhyaya, Achintya K; Krishnan, Kathiresan; Taylor, Amanda; Benz, Ann M; Manion, Brad; Evers, Alex S; Covey, Douglas F; Zorumski, Charles F; Mennerick, Steven