Orally Bioavailable and Site-Selective Covalent STING Inhibitor Derived from a Macrocyclic Marine Diterpenoid
一种源自大环海洋二萜类化合物的口服生物利用度高且具有位点选择性的共价STING抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c02665
Guang-Hao Niu ,Wan-Chi Hsiao ,Po-Hsun Lee ,Li-Guo Zheng ,Yu-Shao Yang ,Wei-Cheng Huang ,Chih-Chien Hsieh ,Tai-Yu Chiu ,Jing-Ya Wang ,Ching-Ping Chen ,Chen-Lung Huang ,May-Su You ,Yi-Ping Kuo ,Chien-Ming Wang ,Zhi-Hong Wen ,Guann-Yi Yu ,Chiung-Tong Chen ,Ya-Hui Chi ,Chun-Wei Tung ,Shu-Ching Hsu ,Teng-Kuang Yeh ,Ping-Jyun Sung ,Mingzi M Zhang ,Lun Kelvin Tsou