Discovery of a novel binding pocket in PPARγ for partial agonists: structure-based virtual screening identifies ginsenoside Rg5 as a partial agonist promoting beige adipogenesis.
在 PPARγ 中发现一种新的部分激动剂结合口袋:基于结构的虚拟筛选鉴定出人参皂苷 Rg5 是一种促进米色脂肪生成的部分激动剂
期刊:Frontiers in Chemistry
影响因子:4.2
doi:10.3389/fchem.2025.1579445
Wang Zhen, Shui Kexin, Zhang Zehui, Chen Yihan, Yang Nanfei, Ji Shiliang, Shen Pingping, Tian Qiang