日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pro-Inflammatory Protein PSCA Is Upregulated in Neurological Diseases and Targets β2-Subunit-Containing nAChRs

促炎蛋白PSCA在神经系统疾病中表达上调,并靶向含有β2亚基的nAChRs

Mikhail A Shulepko ,Yuqi Che ,Alexander S Paramonov ,Milita V Kocharovskaya ,Dmitrii S Kulbatskii ,Anisia A Ivanova ,Anton O Chugunov ,Maxim L Bychkov ,Artem V Kirichenko ,Zakhar O Shenkarev ,Mikhail P Kirpichnikov ,Ekaterina N Lyukmanova

MODULATION OF THE DOPAMINERGIC NEUROTRANSMISSION BY CONTROLLING THE ACTIVITY OF TYROSINE HYDROXYLASE

通过控制酪氨酸羟化酶的活性来调节多巴胺能神经传递

Lyukmanova, Ekaterina N; Shulepko, Mikhail A; Buldakova, Svetlana L; Kasheverov, Igor E; Shenkarev, Zakhar O; Reshetnikov, Roman V; Filkin, Sergey Y; Kudryavtsev, Denis S; Ojomoko, Lucy O; Kryukova, Elena V; Dolgikh, Dmitry A; Kirpichnikov, Mikhail P; Bregestovski, Piotr D; Tsetlin, Victor I; Ichinose, *Hiroshi; Aida, Rina; Nago-Iwashita, Yuka; Moriya, Yuki; Ide, Soichiro; Ikeda, Kazutaka

Recombinant Production, SpeciesSpecific Activity at the TRPA1 Channel, and Significance of the N-Terminal Residue of ProTx-I Toxin from Thrixopelma Pruriens Tarantula Venom

重组生产、TRPA1通道的物种特异性活性以及来自刺猬蛛毒液的ProTx-I毒素N端残基的意义

Shulepko, M A; Zhang, M; Zhivov, E A; Kulbatskii, D S; Paramonov, A S; Che, Yu; Kuznetsov, A V; Popov, A V; Kirpichnikov, M P; Shenkarev, Z O; Lyukmanova, E N

Combination with a Low Dose of Doxorubicin Further Boosts the Antitumor Effect of SLURP-1 In Vivo and Associates with EGFR Down-Regulation.

与低剂量阿霉素联合使用可进一步增强 SLURP-1 在体内的抗肿瘤作用,并与 EGFR 下调相关

Shlepova O V, Bychkov M L, Shipunova V O, Shramova E I, Shulepko M A, Gornostaeva T Y, Kiseleva E A, Kukushkin I D, Kazakov V A, Tukhovskaya E A, Dyachenko I A, Murashev A N, Shenkarev Z O, Deyev S M, Kirpichnikov M P, Lyukmanova E N

Upregulation of cholinergic modulators Lypd6 and Lypd6b associated with autism drives anxiety and cognitive decline

与自闭症相关的胆碱能调节因子 Lypd6 和 Lypd6b 的上调会导致焦虑和认知能力下降

Isaev, Aizek B; Bychkov, Maxim L; Kulbatskii, Dmitrii S; Andreev-Andrievskiy, Alexander A; Mashkin, Mikhail A; Shulepko, Mikhail A; Shlepova, Olga V; Loktyushov, Eugene V; Latanov, Alexander V; Kirpichnikov, Mikhail P; Lyukmanova, Ekaterina N

In Search of the Role of Three-Finger Starfish Proteins

寻找三指海星蛋白的作用

Ekaterina N Lyukmanova, Maxim L Bychkov, Andrei M Chernikov, Ilya D Kukushkin, Dmitrii S Kulbatskii, Sergey V Shabelnikov, Mikhail A Shulepko, Ran Zhao, Wenxiao Guo, Mikhail P Kirpichnikov, Zakhar O Shenkarev, Alexander S Paramonov

Selective targeting of α7 nicotinic acetylcholine receptor by synthetic peptide mimicking loop I of human SLURP-1 provides efficient and prolonged therapy of epidermoid carcinoma in vivo

通过模拟人类 SLURP-1 环 I 的合成肽选择性靶向 α7 烟碱乙酰胆碱受体,可在体内有效且长时间治疗表皮样癌

O V Shlepova #, M A Shulepko #, V O Shipunova #, M L Bychkov, I D Kukushkin, I A Chulina, V N Azev, E I Shramova, V A Kazakov, A M Ismailova, Y A Palikova, V A Palikov, E A Kalabina, E A Shaykhutdinova, G A Slashcheva, E A Tukhovskaya, I A Dyachenko, A N Murashev, S M Deyev, M P Kirpichnikov, Z O Sh

Molecular Basis for Mambalgin-2 Interaction with Heterotrimeric α-ENaC/ASIC1a/γ-ENaC Channels in Cancer Cells

Mambalgin-2 与癌细胞中异源三聚体 α-ENaC/ASIC1a/γ-ENaC 通道相互作用的分子基础

Lyukmanova, Ekaterina N; Zaigraev, Maxim M; Kulbatskii, Dmitrii S; Isaev, Aizek B; Kukushkin, Ilya D; Bychkov, Maxim L; Shulepko, Mikhail A; Chugunov, Anton O; Kirpichnikov, Mikhail P

Recombinant Production, NMR Solution Structure, and Membrane Interaction of the Phα1β Toxin, a TRPA1 Modulator from the Brazilian Armed Spider Phoneutria nigriventer

Phα1β 毒素(巴西武装蜘蛛 Phoneutria nigriventer 的一种 TRPA1 调节剂)的重组产生、NMR 溶液结构和膜相互作用

Ekaterina N Lyukmanova, Pavel A Mironov, Dmitrii S Kulbatskii, Mikhail A Shulepko, Alexander S Paramonov, Elizaveta M Chernaya, Yulia A Logashina, Yaroslav A Andreev, Mikhail P Kirpichnikov, Zakhar O Shenkarev

New Three-Finger Protein from Starfish Asteria rubens Shares Structure and Pharmacology with Human Brain Neuromodulator Lynx2

来自海星(Asteria rubens)的新型三指蛋白与人脑神经调节因子 Lynx2 具有相似的结构和药理作用。

Paramonov, Alexander S; Shulepko, Mikhail A; Makhonin, Alexey M; Bychkov, Maxim L; Kulbatskii, Dmitrii S; Chernikov, Andrey M; Myshkin, Mikhail Yu; Shabelnikov, Sergey V; Shenkarev, Zakhar O; Kirpichnikov, Mikhail P; Lyukmanova, Ekaterina N