日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Bioisosteric Replacement of Amides with 1,2,3-Triazoles Improves Dopamine D4 Receptor Ligand Pharmacokinetics

用1,2,3-三唑类化合物生物等排取代酰胺类化合物可改善多巴胺D4受体配体的药代动力学

Alkhatib, Mohammad; Jakobs, Franziska M; Hanson, John N; Nilson, Ashley N; Moritz, Amy E; Li, Tian; Faibille, Afua B; Bourn, Lindsay A; Ramdhan, Peter A; Ricchezza, Joseph 4th; Jordan, Shannon; Panasis, Diandra; Nguyen, Norman; Kasarla, Nitish; Wang, Bryant; Garcia, Sergio Sola; Saez, Julianna; Paule, James; Lee, Chae Bin; Rais, Rana; Slusher, Barbara S; Sibley, David R; Li, Chenglong; Keck, Thomas M; Boateng, Comfort A

Dissociable control of motivation and reinforcement by distinct ventral striatal dopamine receptors.

腹侧纹状体多巴胺受体对动机和强化进行可分离控制

Enriquez-Traba Juan, Arenivar Miguel, Yarur-Castillo Hector E, Noh Chloe, Flores Rodolfo J, Weil Tenley, Roy Snehashis, Usdin Ted B, LaGamma Christina T, Wang Huikun, Tsai Valerie S, Kerspern Damien, Moritz Amy E, Sibley David R, Lutas Andrew, Moratalla Rosario, Freyberg Zachary, Tejeda Hugo A

Discovery, Characterization, and Optimization of a Novel Positive Allosteric Modulator-Antagonist of the D(3) Dopamine Receptor.

发现、表征和优化一种新型的D(3)多巴胺受体正向变构调节剂-拮抗剂

Moritz Amy E, Wang Feijun, Madaras Nora S, Kelley Amber M, Snyder Kirsten K, Gandhi Disha, Inbody Laura R, Akano Emmanuel O, Shi Lei, Lane J Robert, Free R Benjamin, Frankowski Kevin J, Sibley David R

Multiple Allosteric Sites Allow for Synergistic Enhancement of GPCR Signaling

多个变构位点可协同增强GPCR信号传导

Wang, Kai; Dimova, Snezana T; Hanson, John N; Thakur, Abhishek; Xu, Youwei; Liu, Yini; Moritz, Amy E; Goldberg, Alexander; Xie, Bing; Rayadurgam, Jayachandra; Wang, Feijun; Nilson, Ashley N; Luderman, Kathryn D; Free, R Benjamin; Hu, Wen; Zhang, Jian; Xu, H Eric; Frankowski, Kevin J; Wang, Yue; Shi, Lei; Sibley, David R; Zhuang, Youwen

The Enduring Impact of Pharmacological Reviews-Editorial

药理学评论的持久影响——社论

Sibley, David R

Dopamine receptor divergence revealed using a common ligand

利用共同配体揭示多巴胺受体的差异

Sibley, David R; Nilson, Ashley N; Moritz, Amy E; Shi, Lei

Delineation of G Protein-Coupled Receptor Kinase Phosphorylation Sites within the D(1) Dopamine Receptor and Their Roles in Modulating β-Arrestin Binding and Activation

D(1)多巴胺受体内G蛋白偶联受体激酶磷酸化位点的界定及其在调节β-arrestin结合和激活中的作用

Moritz, Amy E; Madaras, Nora S; Rankin, Michele L; Inbody, Laura R; Sibley, David R

Dissociable control of motivation and reinforcement by distinct ventral striatal dopamine receptors

腹侧纹状体多巴胺受体对动机和强化进行可分离的控制

Enriquez-Traba, Juan; Yarur-Castillo, Hector E; Flores, Rodolfo J; Weil, Tenley; Roy, Snehashis; Usdin, Ted B; LaGamma, Christina T; Arenivar, Miguel; Wang, Huikun; Tsai, Valerie S; Moritz, Amy E; Sibley, David R; Moratalla, Rosario; Freyberg, Zachary Z; Tejeda, Hugo A

Time will tell. Reply to "Comments to pharmacological and behavioral divergence of ketamine enantiomers by Jordi Bonaventura et al." by Chen et al

时间会证明一切。回复 Chen 等人对 Jordi Bonaventura 等人“关于氯胺酮对映体药理学和行为学差异的评论”的评论。

Bonaventura, Jordi; Lam, Sherry; Carlton, Meghan; Boehm, Matthew; Gomez, Juan L; Solís, Oscar; Sánchez-Soto, Marta; Morris, Patrick J; Fredriksson, Ida; Thomas, Craig J; Sibley, David R; Shaham, Yavin; Zarate, Carlos A Jr; Michaelides, Michael

Novel Cryo-EM structures of the D1 dopamine receptor unlock its therapeutic potential

D1多巴胺受体的新型冷冻电镜结构揭示了其治疗潜力

Sibley, David R; Luderman, Kathryn D; Free, R Benjamin; Shi, Lei