日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Molecular basis for the activation of Aurora A and Plk1 kinases during mitotic entry.

有丝分裂开始时 Aurora A 和 Plk1 激酶激活的分子基础。

Pillan Anaïs, Ormancey Philippine, Ben Choug Celia, Orlicky Stephen, Tavernier Nicolas, Van Hove Lucie, Ossareh-Nazari Batool, Joly Nicolas, Sicheri Frank, Lorca Thierry, Pintard Lionel

Discovery and development of potent and selective dual NUAK/MARK inhibitors as Hippo pathway modulators for the treatment of cancer

发现和开发高效且选择性的双重NUAK/MARK抑制剂,作为Hippo通路调节剂用于癌症治疗

Smil, David; Liu, Yong; Xin, Tao; Kiyota, Taira; Aman, Ahmed; Grouleff, Julie; Hoffer, Laurent; Joshi, Dhananjay C; Inanlou, Mohammad R; Song, Siyuan; Mao, Daniel Y L; Ogunjimi, Abiodun A; Pau, Victor; Chini, Fiona D; Kurinov, Igor; Zhang, Ying; Nguyen, Anh Thu; Wrana, Jeffrey L; Sicheri, Frank; Attisano, Liliana; Uehling, David; Al-Awar, Rima; Isaac, Methvin B

A Chemical-Genetic Interaction Matrix Reveals Drug Mechanism and Genetic Architecture

化学-遗传相互作用矩阵揭示药物机制和遗传结构

Coulombe-Huntington, Jasmin; Bertomeu, Thierry; Huard, Caroline; Chatr-Aryamontri, Andrew; St-Cyr, Daniel J; Sánchez-Osuna, María; Papadopoli, David; Normandin, Karine; Paydar, Mohammadjavad; McLaughlan, Shannon; St-Denis, Corinne; Zhang, Li; Say, Henry; Palou, Roger; Stark, Chris; Breitkreutz, Bobby-Joe; van der Sloot, Almer M; Manohar, Sandhya; Lavoie, Hugo; Borden, Katherine L B; Raught, Brian; D'Amours, Damien; Sicheri, Frank; Verreault, Alain; Mader, Sylvie; Meloche, Sylvain; Therrien, Marc; Thibault, Pierre; Wilhelm, Brian; Dirks, Peter B; Aitchison, John D; Patton, Elizabeth; King, Randall W; Roux, Philippe P; Sauvageau, Guy; Hoang, Trang; Marinier, Anne; Harrington, Lea; Kwok, Benjamin; Archambault, Vincent; Topisirovic, Ivan; Tyers, Mike

Author Correction: A substrate binding model for the KEOPS tRNA modifying complex

作者更正:KEOPS tRNA修饰复合物的底物结合模型

Beenstock, Jonah; Ona, Samara Mishelle; Porat, Jennifer; Orlicky, Stephen; Wan, Leo C K; Ceccarelli, Derek F; Maisonneuve, Pierre; Szilard, Rachel K; Yin, Zhe; Setiaputra, Dheva; Mao, Daniel Y L; Khan, Morgan; Raval, Shaunak; Schriemer, David C; Bayfield, Mark A; Durocher, Daniel; Sicheri, Frank

Author Correction: Structures of KEOPS bound to tRNA reveal functional roles of the kinase Bud32

作者更正:KEOPS与tRNA结合的结构揭示了激酶Bud32的功能作用

Chuquimarca, Samara Mishelle Ona; Beenstock, Jonah; Daou, Salima; Porat, Jennifer; Keszei, Alexander F A; Yin, Jay Z; Beschauner, Tobias; Bayfield, Mark A; Mazhab-Jafari, Mohammad T; Sicheri, Frank

WEE1 inhibitors trigger GCN2-mediated activation of the integrated stress response.

WEE1 抑制剂触发 GCN2 介导的整合应激反应的激活。

Tjeerdsma Rinskje B, Ng Timothy F, Roorda Maurits, Bianchi Daniëlle, Yang Sora, Bonnet Clara, VanInsberghe Michael, Everts Marieke, Bakker Femke J, de Boer H Rudolf, Moatti Nathalie, Hustedt Nicole, Yin Jay Z, Hoeg Lisa, Leibovitch Matthew, Sicheri Frank, van Oudenaarden Alexander, de Jong Steven, van den Berg Jeroen, Tanenbaum Marvin E, Brummelkamp Thijn R, Durocher Daniel, van Vugt Marcel A T M

Molecular glues that inhibit deubiquitylase activity and inflammatory signaling.

抑制去泛素化酶活性和炎症信号的分子胶

Chandler Francesca, Reddy Poli Adi Narayana, Bhutda Smita, Ross Rebecca L, Datta Arindam, Walden Miriam, Walker Kieran, Di Donato Stefano, Cassel Joel A, Prakesch Michael A, Aman Ahmed, Datti Alessandro, Campbell Lisa J, Foglizzo Martina, Bell Lillie, Stein Daniel N, Ault James R, Al-Awar Rima S, Calabrese Antonio N, Sicheri Frank, Del Galdo Francesco, Salvino Joseph M, Greenberg Roger A, Zeqiraj Elton

Analysis of Fbox substrate adapter proteins using ProteoSync, a program for projection of evolutionary conservation onto protein atomic coordinates

利用ProteoSync(一种将进化保守性投影到蛋白质原子坐标上的程序)分析Fbox底物衔接蛋白

Sicheri, Elliot; Mao, Daniel; Tyers, Michael; Sicheri, Frank

FAM72A promotes UNG2 degradation and mutagenesis in human cancer cells.

FAM72A促进人类癌细胞中UNG2的降解和突变

Feng Yuqing, Barbulescu Philip, Chana Chetan K, Shirdarreh Melika, Yang Hong, Wu Lizhen, Mamand Sami, Kashem Mohammad, Zia Amin, Han Ming, Tsao Julissa, Pugh Trevor, Cescon David, Schatz David G, Sicheri Frank, Martin Alberto, Pezo Rossanna C

Phosphorylation as a candidate regulatory mechanism for effector recruitment to tankyrase

磷酸化作为效应分子募集至tankyrase的候选调控机制

Broadway, Benjamin J; Pollock, Katie; Cronin, Nora; Rottapel, Robert; Sicheri, Frank; Guettler, Sebastian