日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

E2 variants for probing E3 ubiquitin ligase activities

用于探测E3泛素连接酶活性的E2变体

Du, Jiale; Andree, Gisele A; Horn-Ghetko, Daniel; Stier, Luca; Singh, Jaspal; Kostrhon, Sebastian; Kiss, Leo; Mann, Matthias; Sidhu, Sachdev S; Schulman, Brenda A

Tetravalent antibodies are more potent and efficacious erythropoiesis-stimulating agents than erythropoietin in vivo.

四价抗体在体内比促红细胞生成素更有效、更强效的促红细胞生成剂。

Adams Jarrett J, Blazer Levi L, Chung Jacky, Karimi Minoo, Davidson Taylor, Blair Bailey, Waddle Carlos, Hokanson Craig A, Bruce Heather A, Singer Alexander U, Tombak Eva-Maria, Gildemann Kiira, Tamberg Nele, Kiiver Kaja, Ustav Mart Jr, Ma Yue, Colombo Luigi, Huang Lily Jun-Shen, Michnick Stephen W, Moe Orson W, Sidhu Sachdev S

Structural Basis of Serine Protease Inhibition by Antibodies from Biased Fab Phage-Display Libraries

偏向性Fab噬菌体展示文库抗体抑制丝氨酸蛋白酶的结构基础

Anderson, Kyle J; Lee, Melody S; Sevillano, Natalia; Chen, Gang; Hornsby, Michael J; Sidhu, Sachdev S; Craik, Charles S

USP10/GSK3β-mediated inhibition of PTEN drives resistance to PI3K inhibitors in breast cancer

USP10/GSK3β介导的PTEN抑制导致乳腺癌对PI3K抑制剂产生耐药性

Kumari, Nishi; Wright, Sarah Ce; Witham, Christopher M; Monserrat, Laia; Palafox, Marta; Richard, John Lc; Costa, Carlotta; Elkabets, Moshe; Agostino, Mark; Klemm, Theresa; Eccles, Melissa; Garnham, Alex; Wu, Ting; Nilsson, Jonas A; Walz, Nikita; Venugopal, Veena; Cerra, Anthony; Vasilevski, Natali; Bridgeman, Stephanie; Bassi, Sona; Saei, Azad; Helal, Moutaz; Neundorf, Philipp; Riedel, Angela; Rosenfeldt, Mathias; Gill, Jespal; Pahor, Nikolett; Hartmann, Oliver; Chung, Jacky; Sidhu, Sachdev S; Moderau, Nina; Jha, Sudhakar; Rodon, Jordi; Diefenbacher, Markus E; Komander, David; Serra, Violeta; Eichhorn, Pieter Johan Adam

Locking CBL TKBD in its native conformation presents a novel therapeutic opportunity in mutant CBL-dependent leukemia.

将 CBL TKBD 锁定在其天然构象中,为突变型 CBL 依赖性白血病提供了一种新的治疗机会

Ahmed Syed Feroj, Anand Jayanthi, Zhang Wei, Buetow Lori, Rishi Loveena, Mitchell Louise, Bohlen Jonathan, Lilla Sergio, Sibbet Gary J, Nixon Colin, Patel Amrita, Majorek Karolina A, Zanivan Sara, Bustamante Jacinta C, Sidhu Sachdev S, Blyth Karen, Huang Danny T

Synthetic antibodies targeting EphA2 induce diverse signaling-competent clusters with differential activation.

靶向 EphA2 的合成抗体可诱导具有不同激活方式的多种信号传导活性簇

Adams Jarrett J, Bruce Heather A, Subramania Suryasree, Ploder Lynda, Garcia Julia, Pot Isabelle, Blazer Levi L, Singer Alexander U, Sidhu Sachdev S

Molecular characterization of a synthetic neutralizing antibody targeting p67 of Theileria parva.

对靶向泰勒虫 p67 的合成中和抗体进行分子表征

Miersch Shane, Singer Alex U, Chen Chao, Fellouse Fred, Gopalsamy Anupriya, Costa Luciano Silva E, Lacasta Anna, Chege Hannah, Chege Naomi, Nene Vishvanath, Sidhu Sachdev S

An asymmetric tetrabody is a potent and efficacious agonist of the erythropoietin receptor in vitro and in vivo.

不对称四抗体是体外和体内促红细胞生成素受体的强效激动剂

Adams Jarrett J, Blazer Levi L, Chung Jacky, Karimi Minoo, Davidson Taylor, Bruce Heather A, Singer Alexander U, Yang Ning, Cardarelli Lia, Pot Isabelle, Colombo Luigi, Huang Lily Jun-Shen, Ma Yue, Michnick Stephen W, Moe Orson W, Sidhu Sachdev S

Effective imaging and treatment of Acute Myeloid Leukemia with radiotheranostics targeting the activated conformation of integrin-βeta2

利用靶向整合素β2活化构象的放射诊断技术,可有效成像和治疗急性髓系白血病

Wadhwa, Anju; Johnson, Haley; Bobba, Kondapa Naidu; Bidkar, Anil P; Mayne, Ellis; Rampersaud, Sham; Mandal, Kamal; Barpanda, Abhilash; Prudhvi, Sanjana; Kang, Amrik S; Greenland, Nancy; Balitzer, Dana; Peter, Robin; Raveendran, Athira; Naik, Shubhankar; Basak, Megha; Kasap, Corynn; Werner, Juwita; López-Álvarez, Marina; Lee, Sang Hee; Steri, Veronica; Adams, Jarret J; Sidhu, Sachdev S; Wilson, David M; Seo, Youngho; VanBrocklin, Henry F; Logan, Aaron C; Wiita, Arun P; Flavell, Robert R

Antigen-binding fragments with improved crystal lattice packing and enhanced conformational flexibility at the elbow region as crystallization chaperones

具有改进的晶格堆积和增强的肘部构象灵活性的抗原结合片段作为结晶伴侣

Bruce, Heather A; Singer, Alexander U; Blazer, Levi L; Luu, Khanh; Ploder, Lynda; Pavlenco, Alevtina; Kurinov, Igor; Adams, Jarrett J; Sidhu, Sachdev S