日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Antimalarial Dibenzannulated Medium-Ring Keto Lactams

抗疟疾二苯并环中环酮内酰胺类药物

Ren, Rongguo; Wang, Xiaofang; Leas, Derek A; Scheurer, Christian; Hoevel, Sarah; Cal, Monica; Chen, Gong; Zhong, Longjin; Katneni, Kasiram; Pham, Thao; Patil, Rahul; Sil, Diptesh; Walters, Matthias J; Schulze, Thomas T; Neville, Andrew J; Dong, Yuxiang; Wittlin, Sergio; Kaiser, Marcel; Davis, Paul H; Charman, Susan A; Vennerstrom, Jonathan L

Determinants of activity at human Toll-like receptors 7 and 8: quantitative structure-activity relationship (QSAR) of diverse heterocyclic scaffolds.

人类 Toll 样受体 7 和 8 的活性决定因素:多种杂环骨架的定量构效关系 (QSAR)

Yoo Euna, Salunke Deepak B, Sil Diptesh, Guo Xiaoqiang, Salyer Alex C D, Hermanson Alec R, Kumar Manoj, Malladi Subbalakshmi S, Balakrishna Rajalakshmi, Thompson Ward H, Tanji Hiromi, Ohto Umeharu, Shimizu Toshiyuki, David Sunil A

Structure-based design of novel human Toll-like receptor 8 agonists

基于结构的新型人Toll样受体8激动剂设计

Kokatla, Hari Prasad; Sil, Diptesh; Tanji, Hiromi; Ohto, Umeharu; Malladi, Subbalakshmi S; Fox, Lauren M; Shimizu, Toshiyoki; David, Sunil A

Toll-like receptor-8 agonistic activities in C2, C4, and C8 modified thiazolo[4,5-c]quinolines.

C2、C4 和 C8 修饰的噻唑并[4,5-c]喹啉类化合物的 Toll 样受体-8 激动活性

Kokatla Hari Prasad, Yoo Euna, Salunke Deepak B, Sil Diptesh, Ng Cameron F, Balakrishna Rajalakshmi, Malladi Subbalakshmi S, Fox Lauren M, David Sunil A

Structure-activity relationships of lipopolysaccharide sequestration in N-alkylpolyamines

N-烷基多胺中脂多糖螯合的构效关系

Shrestha, Anurupa; Sil, Diptesh; Malladi, Subbalakshmi S; Warshakoon, Hemamali J; David, Sunil A