Novel 3-Sulfonamide Dual-Tail Pyrrol-2-one Bridged Molecules as Potent Human Carbonic Anhydrase Isoform Inhibitors: Design, Synthesis, Molecular Modeling Investigation, and Anticancer Activity in MeWo, SK-BR-3, and MG-63 Cell Lines
新型3-磺酰胺双尾吡咯-2-酮桥联分子作为强效人碳酸酐酶同工酶抑制剂:设计、合成、分子建模研究及在MeWo、SK-BR-3和MG-63细胞系中的抗癌活性
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c02586
Al-Matarneh, Cristina M; Simionescu, Natalia; Nicolescu, Alina; Silion, Mihaela; Angeli, Andrea; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola; Pinteala, Mariana; Supuran, Claudiu T