日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Crystal structure of Schistosoma mansoni cathepsin D1 in complex with a nanobody reveals the conformation of the propeptide-bound state

曼氏血吸虫组织蛋白酶D1与纳米抗体复合物的晶体结构揭示了前肽结合状态的构象

Parker, Kelly L; Clarke, John D; Liu, Xiaojiao; Gomes, Barbara F; Eyssen, Lauren E A; Furnham, Nicholas; Paes Silva-Jr, Floriano; Owens, Raymond J

Discovery of [1,2,4]triazolo[1,5-a]pyrimidine-Imatinib Hybrids With Selective Cytotoxic Activity: A Mechanistically Divergent Series From Direct BCR-ABL1 Inhibition

发现具有选择性细胞毒活性的[1,2,4]三唑并[1,5-a]嘧啶-伊马替尼杂合物:与直接抑制BCR-ABL1机制不同的系列

Moura, Stefany Castro Bazan; de Oliveira, Andressa Paula; Neto, Joao de Mello Rezende; Dantas, Rafael Ferreira; Silva-Jr, Floriano Paes; Pimentel, Luiz Claudio; Carvalho, Mayara Salles do Nascimento; Leite, Debora Inacio; da Silva, Daiane Vitoria; Bastos, Monica Macedo; Boechat, Nubia

Workflow for Crystallographic Fragment Screening by Crystal Soaking for Protein Targets: A Case Study on Thioredoxin Glutathione Reductase From Schistosoma mansoni

利用晶体浸泡法筛选蛋白质靶标的晶体学片段的工作流程:以曼氏血吸虫硫氧还蛋白谷胱甘肽还原酶为例

Neto, Lauro R S; Montoya, Bogar O; Brandão-Neto, José; Parker, Kelly; Von Delft, Frank; Furnham, Nicholas; Owens, Raymond J; Silva-Jr, Floriano P

FioSchisto's expert perspective on implementing WHO guidelines for schistosomiasis control and transmission elimination in Brazil

FioSchisto就巴西实施世卫组织血吸虫病控制和消除传播指南的专家观点

Menezes, Camilla Almeida; Montresor, Langia Colli; Jangola, Soraya Torres Gaze; de Mattos, Aline Carvalho; Domingues, Ana Lúcia Coutinho; Júnior, Arnaldo Maldonado; Silva, Clélia Christina Mello; Barbosa, Constança Simões; de Mendonça, Cristiane Lafetá Furtado; Massara, Cristiano Lara; Fonseca, Cristina Toscano; de Oliveira, Edward José; Gomes, Elainne Christine de Souza; da Silva, Elizângela Feitosa; Bezerra, Fernando Schemelzer de Moraes; Silva-Jr, Floriano Paes; de Siqueira, Isadora Cristina; Silva, José Roberto Machado E; Heller, Leo; Farias, Leonardo Paiva; Beck, Lilian C Nobrega Holsbach; Santos, Mariana Cristina Silva; Lima, Mariana Gomes; Mourão, Marina de Moraes; Enk, Martin Johannes; Fernandez, Monica Ammon; Katz, Naftale; Carvalho, Omar Dos Santos; Parreiras, Patrícia Martins; Neves, Renata Heisler; Gava, Sandra Grossi; de Oliveira, Sheilla Andrade; Thiengo, Silvana Carvalho; Favre, Tereza Cristina; Graeff-Teixeira, Carlos; Pieri, Otávio Sarmento; Caldeira, Roberta Lima; da Silva-Pereira, Rosiane A; Rocha, Roberto Sena; Oliveira, Ricardo Riccio

New Imatinib Derivatives with Antiproliferative Activity against A549 and K562 Cancer Cells.

具有抗A549和K562癌细胞增殖活性的新型伊马替尼衍生物

Oliveira Andressa, Moura Stefany, Pimentel Luiz, Neto João, Dantas Rafael, Silva-Jr Floriano, Bastos Monica, Boechat Nubia

Editorial: Current approaches in infectious disease drug discovery

社论:传染病药物研发的最新进展

Silva-Jr, Floriano P; Panda, Siva S; Andrade, Carolina Horta; Furnham, Nicholas

De novo design and bioactivity prediction of SARS-CoV-2 main protease inhibitors using recurrent neural network-based transfer learning

利用基于循环神经网络的迁移学习方法,从头设计并预测SARS-CoV-2主要蛋白酶抑制剂的生物活性

Santana, Marcos V S; Silva-Jr, Floriano P

The diverse mechanisms and anticancer potential of naphthoquinones

萘醌的多种作用机制及其抗癌潜力

Pereyra, Carolina Escardó; Dantas, Rafael Ferreira; Ferreira, Sabrina Baptista; Gomes, Luciano Pinho; Silva-Jr, Floriano Paes

FindTargetsWEB: A User-Friendly Tool for Identification of Potential Therapeutic Targets in Metabolic Networks of Bacteria

FindTargetsWEB:一款用于识别细菌代谢网络中潜在治疗靶点的用户友好型工具

Merigueti, Thiago Castanheira; Carneiro, Marcia Weber; Carvalho-Assef, Ana Paula D'A; Silva-Jr, Floriano Paes; da Silva, Fabricio Alves Barbosa