日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer.

基于结构的Hsp90/HDAC6双重抑制剂的发现及其在侵袭性前列腺癌中的应用

Citarella Andrea, Belluti Silvia, Bonanni Davide, Moi Davide, Piccinini Isabella, Rinaldi Arianna, Papulino Chiara, Benedetti Rosaria, Cuoghi Laura, Ciolo Stefano Di, Silvani Alessandra, Altucci Lucia, Pinzi Luca, Franchini Silvia, Passarella Daniele, Sorbi Claudia, Giannini Clelia, Imbriano Carol, Rastelli Giulio

Sustainable Synthesis of 1,2,3-Triazoles using Cyrene as a Biodegradable Solvent in Click Chemistry

利用环己烯作为可生物降解溶剂,在点击化学中可持续合成1,2,3-三唑

Citarella, Andrea; Fiori, Alessandro; Silvani, Alessandra; Passarella, Daniele; Fasano, Valerio

Nicotinic Acid Derivatives As Novel Noncompetitive α-Amylase and α-Glucosidase Inhibitors for Type 2 Diabetes Treatment

烟酸衍生物作为新型非竞争性α-淀粉酶和α-葡萄糖苷酶抑制剂用于2型糖尿病治疗

Citarella, Andrea; Cavinato, Miriam; Rosini, Elena; Shehi, Haidi; Ballabio, Federico; Camilloni, Carlo; Fasano, Valerio; Silvani, Alessandra; Passarella, Daniele; Pollegioni, Loredano; Nardini, Marco

Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 M(pro) Inhibitors

β-氨基硼酸作为SARS-CoV-2 M(pro)抑制剂的计算设计、合成和生物物理评价

Fassi, Enrico M A; Manenti, Marco; Citarella, Andrea; Dei Cas, Michele; Casati, Sara; Micale, Nicola; Schirmeister, Tanja; Roda, Gabriella; Silvani, Alessandra; Grazioso, Giovanni

Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 M(pro)

发现一种新型三氟甲基重氮丙烯类SARS-CoV-2 M(pro)抑制剂

Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Passarella, Daniele; Giannini, Clelia

Enantiopure β-isocyano-boronic esters: synthesis and exploitation in isocyanide-based multicomponent reactions

对映体纯的β-异氰基硼酸酯:合成及其在异氰化物基多组分反应中的应用

Manenti, Marco; Gusmini, Simone; Lo Presti, Leonardo; Molteni, Giorgio; Silvani, Alessandra

Unexpected chiral vicinal tetrasubstituted diamines via borylcopper-mediated homocoupling of isatin imines

通过硼铜介导的靛红亚胺均偶联反应,意外地合成了手性邻位四取代二胺

Manenti, Marco; Lo Presti, Leonardo; Molteni, Giorgio; Silvani, Alessandra

Isonitrile-Based Multicomponent Synthesis of β-Amino Boronic Acids as β-Lactamase Inhibitors

异腈基多组分合成β-氨基硼酸作为β-内酰胺酶抑制剂

Bassini, Emanuele; Gazzotti, Stefano; Sannio, Filomena; Presti, Leonardo Lo; Sgrignani, Jacopo; Docquier, Jean-Denis; Grazioso, Giovanni; Silvani, Alessandra

One step access to oxindole-based β-lactams through Ugi four-center three-component reaction

通过Ugi四中心三组分反应一步合成基于吲哚的β-内酰胺类化合物

Rainoldi, Giulia; Lesma, Giordano; Picozzi, Claudia; Lo Presti, Leonardo; Silvani, Alessandra

Heteronanoparticles by Self-Assembly of Ecdysteroid and Doxorubicin Conjugates To Overcome Cancer Resistance

利用蜕皮甾类激素和阿霉素缀合物的自组装制备异质纳米颗粒以克服癌症耐药性

Fumagalli, Gaia; Giorgi, Giulia; Vágvölgyi, Máté; Colombo, Eleonora; Christodoulou, Michael S; Collico, Veronica; Prosperi, Davide; Dosio, Franco; Hunyadi, Attila; Montopoli, Monica; Hyeraci, Mariafrancesca; Silvani, Alessandra; Lesma, Giordano; Via, Lisa Dalla; Passarella, Daniele