Structural and Atropisomeric Factors Governing the Selectivity of Pyrimido-benzodiazipinones as Inhibitors of Kinases and Bromodomains
嘧啶并苯并二嗪酮作为激酶和溴结构域抑制剂的选择性受结构和阻转异构体因素的影响
期刊:ACS Chemical Biology
影响因子:3.8
doi:10.1021/acschembio.7b00638
Wang, Jinhua; Erazo, Tatiana; Ferguson, Fleur M; Buckley, Dennis L; Gomez, Nestor; Muñoz-Guardiola, Pau; Diéguez-Martínez, Nora; Deng, Xianming; Hao, Mingfeng; Massefski, Walter; Fedorov, Oleg; Offei-Addo, Nana Kwaku; Park, Paul M; Dai, Lingling; DiBona, Amy; Becht, Kelly; Kim, Nam Doo; McKeown, Michael R; Roberts, Justin M; Zhang, Jinwei; Sim, Taebo; Alessi, Dario R; Bradner, James E; Lizcano, Jose M; Blacklow, Stephen C; Qi, Jun; Xu, Xiang; Gray, Nathanael S