日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting autophagy impairment improves the phenotype of a novel CLN8 zebrafish model

针对自噬损伤可改善新型 CLN8 斑马鱼模型的表型

Maria Marchese, Sara Bernardi, Asahi Ogi, Rosario Licitra, Giada Silvi, Serena Mero, Daniele Galatolo, Nicola Gammaldi, Stefano Doccini, Gian Michele Ratto, Simona Rapposelli, Stephan C F Neuhauss, Jingjing Zang, Silvia Rocchiccioli, Elena Michelucci, Elisa Ceccherini, Filippo M Santorelli

Potential use of TG68 - A novel thyromimetic - for the treatment of non-alcoholic fatty liver (NAFLD)-associated hepatocarcinogenesis

TG68(一种新型拟甲状腺素药物)在治疗非酒精性脂肪肝 (NAFLD) 相关肝癌方面的潜在用途

Andrea Caddeo, Marina Serra, Francesca Sedda, Andrea Bacci, Clementina Manera, Simona Rapposelli, Amedeo Columbano, Andrea Perra, Marta Anna Kowalik

New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2

对 2 型大麻素受体双位正构/变构配体的新见解

Rebecca Ferrisi, Beatrice Polini, Caterina Ricardi, Francesca Gado, Kawthar A Mohamed, Giovanna Baron, Salvatore Faiella, Giulio Poli, Simona Rapposelli, Giuseppe Saccomanni, Giancarlo Aldini, Grazia Chiellini, Robert B Laprairie, Clementina Manera, Gabriella Ortore

Synthetic Thyroid Hormone Receptor-β Agonists Promote Oligodendrocyte Precursor Cell Differentiation in the Presence of Inflammatory Challenges

合成甲状腺激素受体-β 激动剂在炎症刺激下促进少突胶质细胞前体细胞分化

Vito Antonio Baldassarro, Corinne Quadalti, Massimiliano Runfola, Clementina Manera, Simona Rapposelli, Laura Calzà

Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: from Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands

新型 CB2 受体配体的设计、合成和生物活性:从正构和变构调节剂到双立体/双位配体

Francesca Gado, Rebecca Ferrisi, Beatrice Polini, Kawthar A Mohamed, Caterina Ricardi, Elena Lucarini, Sara Carpi, Federica Domenichini, Lesley A Stevenson, Simona Rapposelli, Giuseppe Saccomanni, Paola Nieri, Gabriella Ortore, Roger G Pertwee, Carla Ghelardini, Lorenzo Di Cesare Mannelli, Grazia Ch

Synthesis and In Vitro Characterization of Selective Cannabinoid CB2 Receptor Agonists: Biological Evaluation against Neuroblastoma Cancer Cells

选择性大麻素 CB2 受体激动剂的合成及体外表征:针对神经母细胞瘤癌细胞的生物学评价

Francesca Gado, Rebecca Ferrisi, Sarah Di Somma, Fabiana Napolitano, Kawthar A Mohamed, Lesley A Stevenson, Simona Rapposelli, Giuseppe Saccomanni, Giuseppe Portella, Roger G Pertwee, Robert B Laprairie, Anna Maria Malfitano, Clementina Manera

Design, synthesis and biological evaluation of novel orthosteric-allosteric ligands of the cannabinoid receptor type 2 (CB2R)

大麻素受体 2 型(CB2R)新型正构-变构配体的设计、合成及生物学评价

Rebecca Ferrisi, Francesca Gado, Beatrice Polini, Caterina Ricardi, Kawthar A Mohamed, Lesley A Stevenson, Gabriella Ortore, Simona Rapposelli, Giuseppe Saccomanni, Roger G Pertwee, Robert B Laprairie, Clementina Manera, Grazia Chiellini

Design, Synthesis, and In Vitro Evaluation of Novel 8-Amino-Quinoline Combined with Natural Antioxidant Acids

新型 8-氨基喹啉与天然抗氧化酸结合的设计、合成及体外评价

Andrea Bacci, Francesca Corsi, Massimiliano Runfola, Simona Sestito, Ilaria Piano, Clementina Manera, Giuseppe Saccomanni, Claudia Gargini, Simona Rapposelli

Beyond Antioxidant Effects: Nature-Based Templates Unveil New Strategies for Neurodegenerative Diseases

超越抗氧化作用:基于自然的模板揭示神经退行性疾病的新策略

Bacci, Andrea; Runfola, Massimiliano; Sestito, Simona; Rapposelli, Simona

Chitosan nanoparticles as a promising tool in nanomedicine with particular emphasis on oncological treatment

壳聚糖纳米颗粒作为一种很有前景的纳米医学工具,尤其是在肿瘤治疗领域。

Sharifi-Rad, Javad; Quispe, Cristina; Butnariu, Monica; Rotariu, Lia Sanda; Sytar, Oksana; Sestito, Simona; Rapposelli, Simona; Akram, Muhammad; Iqbal, Mehwish; Krishna, Akash; Kumar, Nanjangud Venkatesh Anil; Braga, Susana S; Cardoso, Susana M; Jafernik, Karolina; Ekiert, Halina; Cruz-Martins, Natália; Szopa, Agnieszka; Villagran, Marcelo; Mardones, Lorena; Martorell, Miquel; Docea, Anca Oana; Calina, Daniela